Target Details
| UniProt AC | Q13188 |
|---|---|
| Gene Symbol | STK3 |
| Protein Name | Serine/threonine-protein kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11629 (Mst1_SARAH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 285
- Clinical molecules 27
- Avg pChEMBL 6.72
KEGG Pathways (4)
Active Molecules (285)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DJOLWWBENMZSKJ
|
6.9 | IC50 | 2 | — | |
ZZSBPGIGIUFJRA
|
6.9 | Kd | 46 | — | |
BGYVWFZMYBWCNY
|
6.8 | Ki | 30 | — | |
DQPYZHUAILXFJI
|
6.8 | Ki | 27 | — | |
GUBJNPWVIUFSTR
|
6.8 | Kd | 103 | — | |
GXKYSFQMTTZPGW
|
6.8 | Ki | 7 | — | |
NKGLJTITEFZKAN
|
6.8 | Ki | 35 | — | |
PQNWNVWJXPSZFR
|
6.8 | Ki | 21 | — | |
RQJIDUOCLNMUHR
|
6.8 | Ki | 15 | — | |
VVEGARMQKNYDID
|
6.8 | Ki | 24 | — | |
YEKVTSRZMPLPFK
|
6.8 | Ki | 17 | — | |
ZGDSBEUMPIMXBM
|
6.8 | Ki | 42 | — | |
QSJSVHCOJILSCM
|
6.8 | IC50 | 2 | — | |
PFFIEMXZEROLOA
|
6.8 | IC50 | 2 | — | |
RQJDPSBBHHYXOK
|
6.7 | IC50 | 2 | — | |
MUOUHNBOXJIELS
|
6.7 | IC50 | 3 | — | |
OVLGSAZYDZSQMN
|
6.7 | IC50 | 2 | — | |
CNQGNADBGYCKKV
|
6.7 | Ki | 25 | — | |
DKSNLQYRZJKYOC
|
6.7 | Ki | 51 | — | |
JAMDNXUAYUHJLJ
|
6.7 | Ki | 40 | — | |
JSKUWFIZUALZLX
|
6.7 | Ki | 33 | — | |
KKYPRNBBPBRJQX
|
6.7 | Ki | 40 | — | |
MULNSLQVKKUPJN
|
6.7 | Ki | 41 | — | |
OLUKILHGKRVDCT
|
6.7 | Ki | 44 | Yes | |
TUJUZVJICDSNLY
|
6.7 | Ki | 19 | — | |
QMQJFRBEIOAQNT
|
6.7 | IC50 | 3 | — | |
AFBCNAMQWNEPEP
|
6.7 | IC50 | 2 | — | |
BMGQWWVMWDBQGC
|
6.7 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.7 | Kd | 91 | Yes | |
ZKQLNNVJKSTDGB
|
6.7 | IC50 | 2 | — | |
FZMKVQZVEVRANJ
|
6.7 | IC50 | 2 | — | |
JMAPTHRNJHOVDP
|
6.6 | IC50 | 3 | — | |
OICKVPGRZUWXPB
|
6.6 | IC50 | 3 | — | |
HVELYDDHAUZMMJ
|
6.6 | IC50 | 2 | — | |
NCXSLSJEOUOJBB
|
6.6 | IC50 | 3 | — | |
AUDNGNGLLRZLDR
|
6.6 | Ki | 33 | — | |
CQBBMNXXVMOFCA
|
6.6 | Ki | 39 | — | |
DBXGGXLBTWZXBB
|
6.6 | Ki | 39 | — | |
FDVSOQRNTAPCHB
|
6.6 | Ki | 40 | — | |
GHPFQRTVUDXWCC
|
6.6 | Ki | 35 | — | |
IBPSHHSPUPWXHN
|
6.6 | Ki | 6 | — | |
JPCWMTOYDYYXLS
|
6.6 | Ki | 7 | — | |
KWRXWPRFIUJQBP
|
6.6 | Ki | 25 | — | |
OADRBDVURCEKRP
|
6.6 | Ki | 44 | — | |
QTQUAHGXBLFSCH
|
6.6 | Ki | 10 | — | |
RFBPWKMQWSIPEO
|
6.6 | Ki | 28 | — | |
RYAVJHIPOWNWDE
|
6.6 | Ki | 38 | — | |
SLKCVFPEQGHNSI
|
6.6 | Ki | 29 | — | |
VXYDJXMHISGSDA
|
6.6 | Ki | 59 | — | |
XMGFTZYNTYNOOJ
|
6.6 | Ki | 10 | — |