Target Details
| UniProt AC | Q13188 |
|---|---|
| Gene Symbol | STK3 |
| Protein Name | Serine/threonine-protein kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11629 (Mst1_SARAH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 285
- Clinical molecules 27
- Avg pChEMBL 6.72
KEGG Pathways (4)
Active Molecules (285)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WINHZLLDWRZWRT
|
7.2 | Kd | 201 | Yes | |
JWNPDZNEKVCWMY
|
7.2 | Kd | 57 | Yes | |
KDKUVYLMPJIGKA
|
7.2 | Kd | 91 | Yes | |
AZTMYWWWILJAKW
|
7.2 | Ki | 16 | Yes | |
CHTMRWQLNNRRFJ
|
7.2 | Ki | 70 | — | |
GHPFSYCYZJKVDZ
|
7.2 | Ki | 18 | Yes | |
IAKGNUWZPSPEKU
|
7.2 | Ki | 19 | — | |
KNACLJBHKVSTDL
|
7.2 | Ki | 40 | — | |
NJPWCTYVEJIQBM
|
7.2 | Ki | 72 | — | |
ULHGAQSVFPOUDY
|
7.2 | Ki | 43 | — | |
CTNPALGJUAXMMC
|
7.2 | Kd | 151 | — | |
DKZYXHCYPUVGAF
|
7.2 | Kd | 112 | — | |
AYRVYPOFYQSRNH
|
7.2 | IC50 | 2 | — | |
BHTWDJBVZQBRKP
|
7.1 | IC50 | 4 | — | |
JTSLALYXYSRPGW
|
7.1 | Kd | 8 | — | |
CNTCGRJDUJEUDG
|
7.1 | Ki | 37 | — | |
GDYZFFBMSBDTAA
|
7.1 | Ki | 60 | — | |
KUNZDWIFPOMUOX
|
7.1 | Ki | 36 | — | |
PCQMERRARZKTPW
|
7.1 | Ki | 68 | — | |
UMTWTCVTRDYHQQ
|
7.1 | Ki | 56 | — | |
WDARYLSSWBWVCU
|
7.1 | Ki | 49 | — | |
XOOAAYRIVATZNM
|
7.1 | Ki | 55 | — | |
XUFLBSMTYMFOQH
|
7.1 | Ki | 43 | — | |
YEHCNYAQEBQCCS
|
7.1 | Ki | 74 | — | |
IAYGCINLNONXHY
|
7.1 | Kd | 50 | — | |
ONFLVQULIQDDSN
|
7.0 | IC50 | 3 | — | |
ADLPKFFMGIJZIM
|
7.0 | Ki | 44 | — | |
JTRNNNVASYCTLO
|
7.0 | Ki | 14 | — | |
NCPXFACDZCEIQL
|
7.0 | Ki | 7 | — | |
ORRHVRJUSPCILV
|
7.0 | Ki | 16 | — | |
WINHZLLDWRZWRT
|
7.0 | Ki | 66 | — | |
XBYVOPRDASFDMY
|
7.0 | Ki | 42 | — | |
XNWKXXIGSPPPBH
|
7.0 | Ki | 31 | — | |
LOGJQOUIVKBFGH
|
7.0 | IC50 | 11 | Yes | |
QHWXURVXTQGCOB
|
6.9 | IC50 | 3 | — | |
QWHANLNIEKAAFF
|
6.9 | IC50 | 2 | — | |
SLOIJUIDHUKLRX
|
6.9 | IC50 | 3 | — | |
VQVBIURGGWKQOR
|
6.9 | IC50 | 2 | — | |
BIKYDWLMTPRSQL
|
6.9 | Ki | 50 | — | |
JZTOUVBEZONDKA
|
6.9 | Ki | 80 | — | |
LCHCSKHPVCDXAU
|
6.9 | Ki | 30 | — | |
MVJMMLFMPWITEJ
|
6.9 | Ki | 110 | — | |
OAVGBZOFDPFGPJ
|
6.9 | Ki | 42 | Yes | |
PRRYQINUAIQTFJ
|
6.9 | Ki | 11 | — | |
PSCJSWRVCKUMSL
|
6.9 | Ki | 35 | — | |
RTYJMUXLFRYRBU
|
6.9 | Ki | 35 | — | |
SRUYMJRFVGLQDV
|
6.9 | Ki | 37 | — | |
UVZVWLFSZNPMBS
|
6.9 | Ki | 17 | — | |
XAHJIRNRDAKTEF
|
6.9 | Ki | 18 | — | |
YUOWJICKAJQZLS
|
6.9 | Ki | 35 | — |