Target Details
| UniProt AC | Q13188 |
|---|---|
| Gene Symbol | STK3 |
| Protein Name | Serine/threonine-protein kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11629 (Mst1_SARAH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 285
- Clinical molecules 27
- Avg pChEMBL 6.72
KEGG Pathways (4)
Active Molecules (285)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.7 | Kd | 213 | — | |
HKSZLNNOFSGOKW
|
9.4 | Ki | 118 | — | |
TVUWQDLBEOZVOU
|
8.8 | Ki | 41 | — | |
UIARLYUEJFELEN
|
8.6 | Kd | 289 | Yes | |
HKSZLNNOFSGOKW
|
8.6 | IC50 | 408 | — | |
OSVUGUHRKMMBSE
|
8.5 | Kd | 170 | — | |
KHGPYYFCIAISBU
|
8.5 | Ki | 31 | — | |
ZKLJKKASNXVQBZ
|
8.4 | Ki | 27 | — | |
NXSJMRCTGYTSTK
|
8.2 | Kd | 200 | — | |
SMRWVXLSRJWVBF
|
8.1 | Ki | 25 | — | |
BSFNGHCTZDCQBF
|
7.9 | Ki | 93 | — | |
ULMCFLZUGRSEQA
|
7.9 | Ki | 17 | — | |
WPHKIQPVPYJNAX
|
7.8 | Ki | 81 | — | |
KNARVZUUCLIBGV
|
7.7 | Ki | 33 | — | |
MCCCQFAOMZMZKE
|
7.7 | Ki | 52 | — | |
DPEXRCOBPACFOO
|
7.6 | Ki | 36 | — | |
FONINLXADYUZFI
|
7.6 | Ki | 25 | — | |
ZCCJKVBTHCOISJ
|
7.6 | Ki | 46 | — | |
FLEAYYMORDPWAJ
|
7.5 | Ki | 90 | — | |
LSLPDHNUWRDOGC
|
7.5 | Ki | 25 | — | |
MHCPAORAYMTGCZ
|
7.5 | Ki | 37 | — | |
PLHUMPJXRHMFFR
|
7.5 | Ki | 28 | — | |
QNUKRWAIZMBVCU
|
7.5 | Ki | 46 | — | |
RBXYGQNZRVPDNB
|
7.5 | Ki | 34 | — | |
XHORJSJFHVABEA
|
7.5 | Ki | 49 | — | |
XKZINYYXWJEYEL
|
7.5 | Ki | 37 | — | |
XZXHXSATPCNXJR
|
7.4 | Kd | 165 | Yes | |
YRDHKIFCGOZTGD
|
7.4 | IC50 | 21 | — | |
ADMFLILDQJSEIK
|
7.4 | Ki | 72 | — | |
DASFSPDIWCMVRW
|
7.4 | Ki | 21 | — | |
HOYRWTWZUFFACV
|
7.4 | Ki | 28 | — | |
LACOMQAWPSFXQC
|
7.4 | Ki | 27 | — | |
UOVCGJXDGOGOCZ
|
7.4 | Ki | 59 | — | |
KOZFSFOOLUUIGY
|
7.4 | Kd | 88 | Yes | |
PBCZSGKMGDDXIJ
|
7.3 | Kd | 68 | Yes | |
APPXQUDJLJXULP
|
7.3 | IC50 | 47 | — | |
BQPLWJRDSDNGNE
|
7.3 | Ki | 16 | — | |
FUMCKNCUEAQHCV
|
7.3 | Ki | 103 | — | |
ILUGAYBMBIJXHC
|
7.3 | Ki | 9 | — | |
LPILBMJJRGTKOQ
|
7.3 | Ki | 27 | — | |
OUJZYQBEFNDJQN
|
7.3 | Ki | 71 | — | |
OWFXKTOLFUQPDJ
|
7.3 | Ki | 36 | — | |
PUYIXDDMOUMMRR
|
7.3 | Ki | 27 | — | |
RYYNGWLOYLRZLK
|
7.3 | Ki | 104 | — | |
UGEJLCNSVIVALC
|
7.3 | Ki | 41 | — | |
YQKSNDNARJQAHP
|
7.3 | Ki | 12 | — | |
YWTBGJGMTBHQTM
|
7.3 | Ki | 65 | — | |
ZGGIYFOLDBTZIL
|
7.3 | Ki | 27 | — | |
ZWVZORIKUNOTCS
|
7.3 | Ki | 69 | — | |
VKBFHTIUXUCYRQ
|
7.2 | Ki | 66 | — |