Target Details
| UniProt AC | Q13177 |
|---|---|
| Gene Symbol | PAK2 |
| Protein Name | Serine/threonine-protein kinase PAK 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00786 (PBD) PF00069 (Pkinase) |
Summary
- Multi-target molecules 47
- Clinical molecules 3
- Avg pChEMBL 7.0
KEGG Pathways (11)
Associated Diseases (1)
Active Molecules (47)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KHDMDYBLHAGOQS
|
8.7 | Ki | 2 | — | |
HKSZLNNOFSGOKW
|
8.6 | IC50 | 408 | — | |
HKSZLNNOFSGOKW
|
8.5 | Kd | 213 | — | |
YYLKKYCXAOBSRM
|
8.4 | Kd | 191 | — | |
SNHDCUDTVCJVGD
|
8.3 | Ki | 2 | — | |
QGBBLDRMFCNXMM
|
8.0 | Ki | 2 | — | |
ZBCMHWUFWQFPLV
|
8.0 | IC50 | 9 | — | |
YJZIVGDUWQTSQX
|
7.7 | Ki | 2 | — | |
RAJHPNYKXCHTBA
|
7.4 | Ki | 2 | — | |
QKNBRNSGPNCARD
|
7.4 | IC50 | 9 | — | |
UIARLYUEJFELEN
|
7.4 | Kd | 289 | Yes | |
RYCBSFIKWACFBY
|
7.3 | Ki | 3 | — | |
GUERACYCGKAFOU
|
7.3 | IC50 | 3 | — | |
HISDSBBMGJUNCI
|
7.2 | IC50 | 3 | — | |
FTGUWURNNBVUBC
|
7.2 | IC50 | 3 | — | |
AKBMXDMYBOYBBK
|
7.2 | IC50 | 3 | — | |
GHYZGSZITPRQRZ
|
7.2 | IC50 | 3 | — | |
WFVHHGNMKJUPFM
|
7.1 | IC50 | 3 | — | |
SFNRLFDMFWZHTP
|
7.1 | IC50 | 2 | — | |
JWNPDZNEKVCWMY
|
7.1 | Kd | 57 | Yes | |
KZHMCSYYLVKDCX
|
7.1 | IC50 | 2 | — | |
WFVHHGNMKJUPFM
|
7.0 | IC50 | 3 | — | |
SGUZXWKWTMWMCR
|
6.9 | IC50 | 4 | — | |
PVZRBQHDDWNKDW
|
6.9 | IC50 | 3 | — | |
AAMUKYFUFDUBDC
|
6.8 | IC50 | 3 | — | |
QWFHISYETQDHDU
|
6.8 | IC50 | 3 | — | |
AYCPARAPKDAOEN
|
6.7 | IC50 | 73 | — | |
UEKXGVNKFSFQPH
|
6.7 | IC50 | 3 | — | |
HKJCMFRABFUAJX
|
6.7 | IC50 | 9 | — | |
GTAKUJFUJVMIPM
|
6.6 | IC50 | 3 | — | |
WTEGSNARHOVIJM
|
6.6 | IC50 | 3 | — | |
DTIPYTJPPYYCBX
|
6.6 | IC50 | 3 | — | |
KGPGFQWBCSZGEL
|
6.6 | Kd | 59 | Yes | |
WFVHHGNMKJUPFM
|
6.6 | IC50 | 3 | — | |
MXFNRZNGPALJHJ
|
6.5 | IC50 | 2 | — | |
NCHCHMGQMPWJRZ
|
6.5 | IC50 | 2 | — | |
NHHQJBCNYHBUSI
|
6.5 | Kd | 220 | — | |
OINGHOPGNMYCAB
|
6.4 | Kd | 2 | — | |
OINGHOPGNMYCAB
|
6.4 | Kd | 2 | — | |
UMEIGUHCOYWUSH
|
6.3 | IC50 | 2 | — | |
BMPPDFZFSRZMRS
|
6.3 | IC50 | 2 | — | |
SNYOTOIHSZLIAL
|
6.2 | IC50 | 2 | — | |
WFVHHGNMKJUPFM
|
6.1 | IC50 | 3 | — | |
OINGHOPGNMYCAB
|
6.1 | IC50 | 2 | — | |
CTHCTGQFKJADML
|
6.0 | IC50 | 2 | — | |
GEEQAZJUJDNBFD
|
6.0 | Ki | 2 | — | |
RZXMIHOUHYSGJO
|
6.0 | IC50 | 4 | — |