Target Details
| UniProt AC | Q13164 |
|---|---|
| Gene Symbol | MAPK7 |
| Protein Name | Mitogen-activated protein kinase 7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 46
- Clinical molecules 8
- Avg pChEMBL 6.74
KEGG Pathways (8)
Active Molecules (46)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CBWCJYFVVHOTAZ
|
8.0 | IC50 | 3 | — | |
QXURFIGBRGWPQD
|
7.5 | IC50 | 2 | — | |
OVPNQJVDAFNBDN
|
7.4 | Kd | 44 | Yes | |
VXBAJLGYBMTJCY
|
7.4 | IC50 | 34 | Yes | |
QQWUGDVOUVUTOY
|
7.3 | Kd | 231 | Yes | |
HOMJAAIVTDVQJA
|
7.2 | IC50 | 2 | — | |
VDNUIDRDCANSTA
|
7.2 | IC50 | 2 | — | |
JGVXSQJYBQAPAE
|
7.2 | IC50 | 3 | — | |
JOOXLOJCABQBSG
|
7.2 | Kd | 139 | — | |
NGSRRJBACKDZHY
|
7.1 | IC50 | 3 | — | |
DDTPGANIPBKTNU
|
7.1 | IC50 | 8 | — | |
XDCQYSVFUPULSL
|
7.0 | IC50 | 2 | — | |
YYTFTZONXCQXLW
|
7.0 | IC50 | 3 | — | |
JRNJNYBQQYBCLE
|
7.0 | Kd | 40 | Yes | |
HKSZLNNOFSGOKW
|
6.9 | IC50 | 408 | — | |
HEIWGGHLGABSLB
|
6.9 | Kd | 10 | — | |
GFDDTDKCZCGJLM
|
6.9 | IC50 | 5 | — | |
LIEUQFMVFKJKHX
|
6.8 | IC50 | 10 | — | |
XJNDWYLNOREHCQ
|
6.8 | IC50 | 2 | — | |
NFNBVXVXMQZSGB
|
6.8 | IC50 | 3 | — | |
DXQBCGUEDOHNHP
|
6.8 | Kd | 12 | — | |
OXSKLFUMHBJZNS
|
6.8 | IC50 | 2 | — | |
XVBGRTMNFNMINE
|
6.8 | IC50 | 5 | — | |
UWHQAHZPBAISBU
|
6.7 | IC50 | 2 | — | |
VVPYTOVXFOGRIN
|
6.7 | IC50 | 2 | — | |
QCLXNOBXQUWUEW
|
6.7 | IC50 | 9 | — | |
WWDLVMCJDNTBPK
|
6.7 | IC50 | 3 | — | |
HGHFBVBNHYJNHK
|
6.6 | IC50 | 3 | — | |
YSFFGUHMDPYPAW
|
6.6 | IC50 | 3 | — | |
WUWXJIFZTHONGM
|
6.6 | IC50 | 3 | — | |
ISCJKSNXTHTNBW
|
6.6 | IC50 | 4 | — | |
CRFHZXHUGPCWJA
|
6.5 | IC50 | 8 | — | |
VJDBYVPTQWPRPA
|
6.5 | Kd | 2 | — | |
QRVNXVTYIYXPER
|
6.5 | IC50 | 3 | — | |
XKFTZKGMDDZMJI
|
6.4 | Kd | 64 | Yes | |
DDJBEYRDSUCNLT
|
6.3 | IC50 | 4 | — | |
KTEIFNKAUNYNJU
|
6.3 | Kd | 114 | — | |
KDKUVYLMPJIGKA
|
6.3 | Kd | 91 | Yes | |
BIIVYFLTOXDAOV
|
6.2 | Kd | 29 | — | |
BIIVYFLTOXDAOV
|
6.2 | Kd | 82 | Yes | |
PSPFQEBFYXJZEV
|
6.2 | Kd | 10 | — | |
OUSFTKFNBAZUKL
|
6.2 | Kd | 58 | Yes | |
LGLHCXISMKHLIK
|
6.2 | Kd | 3 | — | |
FSZPIAXLCCQFCM
|
6.1 | IC50 | 2 | — | |
LOYSOCNFHOPWJA
|
6.1 | IC50 | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — |