Target Details
| UniProt AC | Q13163 |
|---|---|
| Gene Symbol | MAP2K5 |
| Protein Name | Dual specificity mitogen-activated protein kinase kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00564 (PB1) PF00069 (Pkinase) |
Summary
- Multi-target molecules 65
- Clinical molecules 22
- Avg pChEMBL 7.25
KEGG Pathways (5)
Active Molecules (65)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XYFPWWZEPKGCCK
|
6.6 | Kd | 34 | — | |
GCIKSSRWRFVXBI
|
6.6 | Kd | 109 | Yes | |
JOOXLOJCABQBSG
|
6.4 | Kd | 139 | — | |
VYPGLYMWNDRFGZ
|
6.4 | Kd | 12 | — | |
CUIHSIWYWATEQL
|
6.3 | Kd | 61 | Yes | |
OOMBFNDWQIGHEK
|
6.3 | Kd | 22 | — | |
XLSYZSRXVVCHLS
|
6.3 | Kd | 48 | — | |
XGALLCVXEZPNRQ
|
6.2 | Kd | 39 | Yes | |
GMIZZEXBPRLVIV
|
6.2 | Kd | 6 | — | |
GPXBXXGIAQBQNI
|
6.1 | Kd | 11 | — | |
HHCBMISMPSAZBF
|
6.1 | IC50 | 23 | — | |
SUDAHWBOROXANE
|
6.1 | Kd | 6 | — | |
HZRJHVDNTDBTOZ
|
6.1 | IC50 | 8 | — | |
QHUDPFOODLMGQO
|
6.1 | IC50 | 5 | — | |
CSGQVNMSRKWUSH
|
6.0 | Kd | 21 | — |