Target Details
| UniProt AC | Q13163 |
|---|---|
| Gene Symbol | MAP2K5 |
| Protein Name | Dual specificity mitogen-activated protein kinase kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00564 (PB1) PF00069 (Pkinase) |
Summary
- Multi-target molecules 65
- Clinical molecules 22
- Avg pChEMBL 7.25
KEGG Pathways (5)
Active Molecules (65)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YZDJQTHVDDOVHR
|
9.8 | Kd | 23 | — | |
MWKSRKSEWLRPBL
|
9.1 | Kd | 1075 | — | |
HOMJAAIVTDVQJA
|
8.8 | IC50 | 2 | — | |
VDNUIDRDCANSTA
|
8.8 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
8.7 | Kd | 165 | Yes | |
SEJGTFPOEJWEGG
|
8.6 | Kd | 149 | — | |
LIEUQFMVFKJKHX
|
8.6 | Kd | 10 | — | |
QYZOGCMHVIGURT
|
8.6 | Kd | 26 | Yes | |
ZBNZXTGUTAYRHI
|
8.5 | Kd | 102 | Yes | |
FSZPIAXLCCQFCM
|
8.4 | IC50 | 2 | — | |
OATHVDKMFZZHHN
|
8.2 | Kd | 9 | — | |
UIARLYUEJFELEN
|
8.2 | Kd | 289 | Yes | |
MFAQYJIYDMLAIM
|
8.1 | Kd | 130 | Yes | |
SHPFDGWALWEPGS
|
8.1 | Kd | 35 | — | |
UBPYILGKFZZVDX
|
8.1 | Kd | 130 | Yes | |
HKSZLNNOFSGOKW
|
8.0 | IC50 | 408 | — | |
CXQHYVUVSFXTMY
|
7.7 | Kd | 154 | — | |
BWBUPDTUXQDHSX
|
7.6 | IC50 | 5 | — | |
PIQCTGMSNWUMAF
|
7.5 | Kd | 137 | Yes | |
IKENQUDOTQBCJH
|
7.4 | Kd | 18 | — | |
DYNHJHQFHQTFTP
|
7.4 | Kd | 38 | — | |
NHHQJBCNYHBUSI
|
7.4 | Kd | 220 | — | |
WINHZLLDWRZWRT
|
7.3 | Kd | 201 | Yes | |
LOLPPWBBNUVNQZ
|
7.3 | Kd | 97 | Yes | |
PMDAVRLCSZSLRH
|
7.3 | Kd | 13 | — | |
UHTHHESEBZOYNR
|
7.3 | Kd | 66 | Yes | |
ADPWNOVNIYYWDN
|
7.3 | Kd | 2 | — | |
DKZYXHCYPUVGAF
|
7.2 | Kd | 112 | — | |
VAARYSWULJUGST
|
7.2 | Kd | 119 | Yes | |
OMZCMEYTWSXEPZ
|
7.2 | Kd | 43 | Yes | |
JWNPDZNEKVCWMY
|
7.2 | Kd | 57 | Yes | |
ODPGGGTTYSGTGO
|
7.1 | Kd | 153 | — | |
CTNPALGJUAXMMC
|
7.1 | Kd | 151 | — | |
GBJVVSCPOBPEIT
|
7.1 | Kd | 13 | Yes | |
NZJCXRPMZJGVCC
|
7.1 | Kd | 8 | — | |
AAKJLRGGTJKAMG
|
7.0 | Kd | 50 | Yes | |
GUBJNPWVIUFSTR
|
7.0 | Kd | 103 | — | |
YYLKKYCXAOBSRM
|
6.9 | Kd | 191 | — | |
ISPBCAXOSOLFME
|
6.9 | Kd | 11 | — | |
RITAVMQDGBJQJZ
|
6.8 | Kd | 43 | — | |
USVCWSAJUAARAL
|
6.8 | Kd | 8 | — | |
IAYGCINLNONXHY
|
6.8 | Kd | 50 | — | |
JONPTLGCLPUHKH
|
6.8 | Kd | 8 | — | |
DHZKWPMYADCRCR
|
6.8 | IC50 | 4 | — | |
FLBNLJLONKAPLR
|
6.8 | Kd | 31 | — | |
BIIVYFLTOXDAOV
|
6.7 | Kd | 82 | Yes | |
HHZIURLSWUIHRB
|
6.7 | Kd | 57 | Yes | |
MLDQJTXFUGDVEO
|
6.7 | Kd | 85 | Yes | |
QQWUGDVOUVUTOY
|
6.7 | Kd | 231 | Yes | |
ASMLDRAEBPYENO
|
6.6 | IC50 | 10 | — |