Target Details
| UniProt AC | Q13133 |
|---|---|
| Gene Symbol | NR1H3 |
| Protein Name | Oxysterols receptor LXR-alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 422
- Clinical molecules 0
- Avg pChEMBL 7.18
KEGG Pathways (5)
Active Molecules (422)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MVLVWBZCSDBJRB
|
6.1 | IC50 | 2 | — | |
YLJKCCPSAPDTDJ
|
6.1 | IC50 | 2 | — | |
PRDITVHZXOYDTE
|
6.1 | Ki | 2 | — | |
WLDSAWDEZLQZSP
|
6.1 | Ki | 2 | — | |
XBDCCVVGSIGGTL
|
6.1 | IC50 | 2 | — | |
YOBSSBAJFVWQAA
|
6.1 | IC50 | 2 | — | |
NSXAZYXFYXSEQK
|
6.1 | IC50 | 2 | — | |
DYLGLRCPXIXIET
|
6.1 | Ki | 2 | — | |
UZNDKNPMFSVFET
|
6.1 | Ki | 2 | — | |
CSTOAOCVMBEIPA
|
6.1 | Ki | 2 | — | |
DWVNDOKJFPRSRU
|
6.1 | Ki | 2 | — | |
HBRYTPUBFUUNKX
|
6.1 | Ki | 2 | — | |
LWFAXHWAXCYXSZ
|
6.1 | Ki | 2 | — | |
OXFIAOBJWCENMG
|
6.1 | Ki | 2 | — | |
YZWZMPWHXSZLBQ
|
6.1 | Ki | 3 | — | |
ALICKBCBWBIBQP
|
6.0 | Ki | 2 | — | |
SAKQPFIBVKAZMM
|
6.0 | Ki | 2 | — | |
XXHQLZDZSDSOOP
|
6.0 | Ki | 2 | — | |
MVZUVIXDADTQPL
|
6.0 | Ki | 2 | — | |
XZVKGPBWXMHCFG
|
6.0 | Ki | 2 | — | |
DUSQUBZCYLLKHT
|
6.0 | IC50 | 2 | — | |
YOYQINDKUAALSH
|
6.0 | Ki | 3 | — |