Target Details
UniProt ACQ13133
Gene SymbolNR1H3
Protein NameOxysterols receptor LXR-alpha
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00104 (Hormone_recep) PF00105 (zf-C4)
Summary
  • Multi-target molecules 422
  • Clinical molecules 0
  • Avg pChEMBL 7.18
Top Co-occurrence Targets
Active Molecules (422)
InChIKey pChEMBL Type Targets Clinical
FLJYMVVOBYULHJ 6.4 IC50 2
HFGCUOYYZKNQLX 6.4 Ki 2
GBXFIRKYLMIFBA 6.4 IC50 2
HKNRVRUCDFTKQI 6.4 Ki 2
IOUQCKSTQUVCIP 6.4 IC50 2
UZNDKNPMFSVFET 6.4 Ki 2
CQTCWVWUQDCTSG 6.4 IC50 3
QVTVCGSKZXEEPI 6.4 Ki 2
UOUJAFCLXIURMD 6.4 Ki 2
FWLREOYIIBBODP 6.4 Ki 2
RFGMOPNIYZVCFS 6.4 IC50 2
WPUHRYSDQSXTGR 6.4 IC50 2
ZIQOKIRETRSSNJ 6.4 Ki 2
ISUZFVXNJCGBJL 6.4 Ki 2
FMOAGFUWAWYZBQ 6.3 Ki 2
RKGUCTQUPQWZOT 6.3 IC50 2
CKHYMMLNOQQEMV 6.3 IC50 2
JPIHSYRXQLKCID 6.3 IC50 2
YBOVOEBYAFAWAS 6.3 Ki 2
CDLBQZJYZMCUBN 6.3 IC50 2
OKUGPERZNQXECM 6.3 Ki 2
BCYNXJGQHVLDNU 6.3 Ki 2
JMPXRXGCUIOVIQ 6.3 Ki 2
FCQLLWXAPLXYQV 6.3 IC50 2
RLNMZAJKGCKXRV 6.3 IC50 2
YYFFXRNVMLUSIQ 6.3 Ki 2
QQVBOEBRRVCOPV 6.3 Ki 2
DNNYNSPBJXNYMZ 6.3 IC50 2
GPHDHOZJIQGWQC 6.3 Ki 2
JYFOULIZQPAJEL 6.3 Ki 2
VRCMDLDBHFNHBT 6.3 IC50 2
YBSIHBWDBRSCLD 6.3 Ki 2
AIOWJRXDKURKOW 6.3 IC50 2
BHOVYPMEYZFYON 6.3 IC50 2
DKTPGSDKMSCAGJ 6.3 Ki 2
MXMNSPKGWWEDFT 6.2 Ki 2
GZAPSISRDWGGFB 6.2 IC50 5
ATFXXADQEVAPEW 6.2 Ki 2
DRRBJCNZGQGKSK 6.2 IC50 2
NIRYIUZPINDTNT 6.2 Ki 2
YRDLIUCBIUYNLE 6.2 Ki 2
GADXIGHAARSCIO 6.2 IC50 3
PFKXVMUDIKLGOG 6.2 Ki 2
CHCCPPPOKAASRP 6.2 IC50 2
OZKKLFAIQTYTBH 6.2 Ki 2
LUJCWOPVYNTRBQ 6.2 Ki 2
PUFOJDYFCGHZAC 6.2 Ki 2
FJLDUPMMOBCQAG 6.1 Ki 2
IBJHNZQOUGJVCC 6.1 Ki 2
SYPXZIFSIJUYCS 6.1 IC50 5
2D structure