Target Details
UniProt ACQ13133
Gene SymbolNR1H3
Protein NameOxysterols receptor LXR-alpha
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00104 (Hormone_recep) PF00105 (zf-C4)
Summary
  • Multi-target molecules 422
  • Clinical molecules 0
  • Avg pChEMBL 7.18
Top Co-occurrence Targets
Active Molecules (422)
InChIKey pChEMBL Type Targets Clinical
HDZWHJYZJWLTAG 6.7 IC50 2
ZMSACEOQWGFPTA 6.7 Ki 2
JFJHGGFPJWKBFT 6.7 Ki 2
VRLNYADEEBSDKC 6.7 Ki 2
OPEYIXLYURKODO 6.7 Ki 2
LJUJGMRQOWUZEL 6.6 IC50 2
AHSVAMKJVNIBDA 6.6 Ki 2
RPEJMRBNVYJBHP 6.6 Ki 2
CUPCXDRVHZGUGE 6.6 IC50 2
LOFRRPNYSLDHRM 6.6 Ki 2
WWWVODUMLXMIRV 6.6 Ki 2
XQWURCYLMCTAFE 6.6 Ki 3
NHSFDMDEDPAKNH 6.6 IC50 2
PICJKSLPJSZRIV 6.6 Ki 2
IQTBHLOUVIJISQ 6.6 IC50 2
WQLPRQYFFAOTOS 6.6 Ki 2
KXXPROPFBQVDKT 6.6 IC50 2
VLCMRTMCMQJSKM 6.6 IC50 2
YIRPKYOIUDNERT 6.6 Ki 2
AWFKUZKMHLKRBA 6.6 IC50 2
DFAPREYFHSKSRA 6.6 IC50 2
TYSRYKHSEFCGPN 6.6 Ki 2
XRYDEEKHRNPJOZ 6.6 Ki 3
DJSVQYMUGOLIIN 6.6 Ki 2
LWXOLPDIDYBJQJ 6.6 Ki 2
TZRCVICHXMBFCB 6.6 IC50 2
LGRUCHCYEMOENE 6.5 IC50 2
MEBPCMPPKTYENX 6.5 IC50 2
YPGJKBPNUAZVOT 6.5 Ki 2
BYZAOZSASXJAQT 6.5 IC50 2
IEPOYBLCAUUPJP 6.5 IC50 2
RGQJDOMXMZANLJ 6.5 IC50 2
JJUUTJCZMGZJDZ 6.5 Kd 3
LMEZNWUTYWBWHN 6.5 IC50 2
QBUILYGRQMFSAV 6.5 IC50 2
VOOZJAGZCXOELE 6.5 Ki 3
BKPFNLPLHXLDDZ 6.5 IC50 2
CABUZECPUSGGRX 6.5 Ki 2
GEXZSCVAMWWQAV 6.5 Ki 2
GKSVBRSAJNOJOL 6.5 Ki 2
GREUENDQALGMMV 6.5 IC50 2
GWAZQHKDYABFCB 6.5 Ki 2
QGOMJEFGXRFUAA 6.5 IC50 2
KCTVTEAWWHOHNZ 6.4 IC50 2
OBXLHEARDPFUMN 6.4 Ki 2
UATPJWGKTPZRPL 6.4 Ki 2
VJEBBKVWKHODQJ 6.4 IC50 2
FFEMTQPBRTULCE 6.4 IC50 2
NTXMYMGYFCGBAL 6.4 IC50 2
DTDVBYRJYQLMSF 6.4 IC50 2
2D structure