Target Details
UniProt ACQ13133
Gene SymbolNR1H3
Protein NameOxysterols receptor LXR-alpha
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00104 (Hormone_recep) PF00105 (zf-C4)
Summary
  • Multi-target molecules 422
  • Clinical molecules 0
  • Avg pChEMBL 7.18
Top Co-occurrence Targets
Active Molecules (422)
InChIKey pChEMBL Type Targets Clinical
PPAHYKJOKMIXNQ 6.9 IC50 2
HDDKTNCZLILPNB 6.9 Ki 3
HLMVLEINLZPXPH 6.9 Ki 2
ZFAZSJUOGZNAMM 6.9 Ki 2
XQHTVSOMTJRZEI 6.9 Ki 2
YYIDRXGXLIOEDJ 6.8 IC50 2
NTWOSTRWTSTGLC 6.8 Ki 2
PAXOTBRHGNYSDC 6.8 Ki 2
QJGPMJDHZAMQSJ 6.8 Ki 2
RGPYRFIDCPYCJL 6.8 Ki 2
CENYEUAKMJYAFN 6.8 Ki 2
DCFHWWUSMITHJJ 6.8 IC50 2
UVRFHLLVIGMMMM 6.8 Ki 2
YNYIBKWUFCUQQY 6.8 IC50 2
ZXTOKWKHXXGVMT 6.8 Ki 3
HVOUQCTVPWXRRS 6.8 Ki 2
HXOUVMGQDQYWNM 6.8 Ki 2
IDKRBDPKBAQNEZ 6.8 IC50 2
KJPPQVNZYDPQRM 6.8 IC50 2
NRUNDIXYUOKLPO 6.8 Ki 2
AEMSEMKBOULOJG 6.8 Ki 2
BHKSYENPDNOBLX 6.8 IC50 2
VIEODBHSIYUQTK 6.8 Ki 2
FHEOPZZFNWUQEY 6.8 IC50 2
HYFGFUVRQMLYAH 6.8 Ki 2
RPEJMRBNVYJBHP 6.8 Ki 2
FKCNXNPZSKIRIX 6.8 Kd 3
XLYCLDVZZOFLRE 6.8 Ki 2
SYMWSPSNNOTRBN 6.8 Ki 2
KYWWJENKIMRJBI 6.8 IC50 3
STNGIHCHDLCYEV 6.8 Ki 3
GMKDRYOJWQXLTE 6.7 IC50 2
KDKLTCKHENMCSN 6.7 Ki 3
OMMCNHJJHLQJHQ 6.7 Ki 2
YYVCZYRPPBVGDX 6.7 Ki 2
WZDFAJOVHXXHKS 6.7 Ki 2
BKOKGTVPLDCTIS 6.7 Ki 2
CRBFBKFQHKHSNV 6.7 Ki 2
ISXPNMSKZHGGLC 6.7 Ki 2
MQKQOJAXHYOTRU 6.7 Ki 2
WLYJUBOVJNVBDO 6.7 Ki 2
PXRKUDZYCJZQBB 6.7 IC50 2
QSIMLIBNOBVYGV 6.7 IC50 2
SAIJBWDHHOMPIR 6.7 IC50 2
ZJPIFOVRFHBVNC 6.7 IC50 2
DYLLPHYLYLHOKV 6.7 Ki 2
LYILZTQKEIMJDW 6.7 Ki 3
OHDRXCKGYPYQAU 6.7 IC50 2
RZPAXNJLEKLXNO 6.7 Ki 2
GEXZSCVAMWWQAV 6.7 Ki 2
2D structure