Target Details
| UniProt AC | Q13133 |
|---|---|
| Gene Symbol | NR1H3 |
| Protein Name | Oxysterols receptor LXR-alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 422
- Clinical molecules 0
- Avg pChEMBL 7.18
KEGG Pathways (5)
Active Molecules (422)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MYNWRKZLIIDPBU
|
8.2 | IC50 | 2 | — | |
QMAWFUWIOSWDJM
|
8.2 | IC50 | 2 | — | |
XOTHLYNSDMSVGX
|
8.2 | Ki | 2 | — | |
GUEIWDLJEBMFMQ
|
8.1 | IC50 | 2 | — | |
IKEBXOQTSPUHRL
|
8.1 | IC50 | 2 | — | |
LMLSWHPQUWFGHJ
|
8.1 | IC50 | 2 | — | |
AVHJCISEWCJAIL
|
8.1 | IC50 | 2 | — | |
DPAWQSUVLANLRD
|
8.1 | IC50 | 2 | — | |
ZLCICKWEGSYHOX
|
8.1 | IC50 | 2 | — | |
FWTLKBYOKWCAEO
|
8.1 | IC50 | 2 | — | |
ISMQLWMZRUKHEF
|
8.1 | IC50 | 2 | — | |
PDIDLFFWXHKWMR
|
8.1 | IC50 | 2 | — | |
SYTLPMIZCIQSJE
|
8.1 | IC50 | 2 | — | |
UCPCLSOVORSWOU
|
8.1 | IC50 | 2 | — | |
DIEQFJUHAMDHJZ
|
8.1 | IC50 | 2 | — | |
GUQJFTLEMOZJBL
|
8.1 | Ki | 3 | — | |
NVDRYPHMVKODMP
|
8.1 | IC50 | 2 | — | |
NXAQUWGSGCUYGJ
|
8.1 | Ki | 2 | — | |
VCNKBGCNOUBXAD
|
8.1 | Ki | 2 | — | |
VXHRQVMQVYQGQG
|
8.0 | IC50 | 2 | — | |
BKINFWHEJAZZTL
|
8.0 | IC50 | 2 | — | |
GKRQECRQGLCHTJ
|
8.0 | IC50 | 2 | — | |
NKFDLBSCCAQKKW
|
8.0 | IC50 | 2 | — | |
AAXKPQBGHZNCOJ
|
8.0 | IC50 | 2 | — | |
JQOOZVXMCPGTNO
|
8.0 | IC50 | 2 | — | |
WPGIFTVVEKGIGJ
|
8.0 | Ki | 3 | — | |
APHRFSGOWKZUGE
|
7.9 | IC50 | 2 | — | |
GEDMLXRPUQZAAS
|
7.9 | IC50 | 2 | — | |
JRJIJEXVKDFRTL
|
7.9 | IC50 | 2 | — | |
QQNXCYFWSCPJOI
|
7.9 | IC50 | 2 | — | |
FLQMNHODIBPHAJ
|
7.9 | IC50 | 2 | — | |
MVQGOFQHJVGQCO
|
7.9 | IC50 | 2 | — | |
SGIWFELWJPNFDH
|
7.9 | IC50 | 6 | — | |
SNVDXERLZQEYID
|
7.9 | IC50 | 2 | — | |
DHCPTZAZDOXILJ
|
7.9 | IC50 | 2 | — | |
NSWRBHFZGBXSGU
|
7.8 | Ki | 2 | — | |
SYOKLRCUKUPRMN
|
7.8 | IC50 | 2 | — | |
WZXCTCJIJVBAOX
|
7.8 | IC50 | 2 | — | |
SQHRBEDYCPJCNA
|
7.8 | IC50 | 2 | — | |
USWOEXHVBVCJOR
|
7.8 | IC50 | 2 | — | |
LCDRBOYRRKJMEX
|
7.8 | IC50 | 2 | — | |
OEDBWXLEGYGITE
|
7.8 | IC50 | 2 | — | |
QTHAGUHHLRNGTA
|
7.8 | Ki | 3 | — | |
VPVFJCQJGDFRIA
|
7.8 | IC50 | 4 | — | |
YAKODSHNCZYDPB
|
7.8 | IC50 | 2 | — | |
LIKCFBAAJFMUJP
|
7.8 | IC50 | 2 | — | |
NKFCIEVAMLCUCO
|
7.8 | IC50 | 2 | — | |
OSCBEESEHIRILI
|
7.8 | Ki | 3 | — | |
CHDZBJMLJJYFFA
|
7.8 | IC50 | 2 | — | |
AJSJAQQMFKYODQ
|
7.7 | IC50 | 2 | — |