Target Details
| UniProt AC | Q13133 |
|---|---|
| Gene Symbol | NR1H3 |
| Protein Name | Oxysterols receptor LXR-alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 422
- Clinical molecules 0
- Avg pChEMBL 7.18
KEGG Pathways (5)
Active Molecules (422)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GBEWPJJHRRWGJD
|
9.1 | IC50 | 2 | — | |
JQOXVKXWQCMPRP
|
9.1 | IC50 | 2 | — | |
DZOUMAUJJDVJHY
|
9.0 | IC50 | 2 | — | |
ASTLYMNMTDERKI
|
9.0 | IC50 | 2 | — | |
SWIBRLXHJPCKAR
|
9.0 | IC50 | 2 | — | |
ZDUOYBOFMKORCT
|
9.0 | IC50 | 2 | — | |
PBQUJALWEDBRLW
|
9.0 | IC50 | 2 | — | |
XZYFDTYSBRYCCK
|
9.0 | IC50 | 2 | — | |
JWRIUHZELXTXLP
|
8.9 | IC50 | 2 | — | |
MFDLTITVUNIPCT
|
8.9 | IC50 | 2 | — | |
SELLUNCDLWGEEU
|
8.9 | IC50 | 2 | — | |
LJZFYKYOXOCPDD
|
8.8 | IC50 | 2 | — | |
QIEBJBNGMINXIF
|
8.8 | IC50 | 2 | — | |
ZIMHQMXADUASSG
|
8.8 | IC50 | 2 | — | |
BUSFVFJRQBYHBW
|
8.8 | IC50 | 2 | — | |
YYDPUXBLDMRZQE
|
8.7 | IC50 | 2 | — | |
HXANPPNXWQVOEO
|
8.7 | IC50 | 2 | — | |
CBDKGOMYQLDSHF
|
8.7 | IC50 | 2 | — | |
CXSWMXMKWWOTPK
|
8.7 | IC50 | 2 | — | |
OUJQRQRBNRGQTC
|
8.7 | IC50 | 2 | — | |
ZXTASCJKIFSEGC
|
8.7 | IC50 | 2 | — | |
INTBHOCJAASBMR
|
8.6 | IC50 | 2 | — | |
MOQUFKNADUILIJ
|
8.6 | IC50 | 2 | — | |
HRXRTZUZVWAYOB
|
8.6 | IC50 | 2 | — | |
XPWTYUUWBMPVLO
|
8.6 | IC50 | 2 | — | |
DZEKZLIXNYUATR
|
8.6 | IC50 | 2 | — | |
QRIKQMLMSCHVRS
|
8.5 | IC50 | 2 | — | |
SWVQEDYQXWDKTA
|
8.5 | Ki | 2 | — | |
VTSLTFRMYLXJLX
|
8.5 | Ki | 2 | — | |
PLHRETMILCOKED
|
8.5 | IC50 | 2 | — | |
LMTALPSNYCOGGX
|
8.5 | IC50 | 2 | — | |
QQDXQGDFJZPVRX
|
8.5 | IC50 | 2 | — | |
ZSOMYKQAXFPKDY
|
8.4 | IC50 | 2 | — | |
RUVMVDAIZHYFPZ
|
8.4 | IC50 | 2 | — | |
GBFXOJGYUQWRBP
|
8.4 | IC50 | 2 | — | |
NYORNGSRUVZKGU
|
8.4 | IC50 | 2 | — | |
SEUOQSBVNSJTTL
|
8.3 | IC50 | 2 | — | |
DRNWBBRZORIYEI
|
8.3 | IC50 | 2 | — | |
MFLGRDLZNMSORM
|
8.3 | IC50 | 2 | — | |
XMSRNUPVXCPJHV
|
8.3 | IC50 | 2 | — | |
AIZFRFCHCJRXFS
|
8.3 | IC50 | 2 | — | |
ZMLDZMJEIPYMEJ
|
8.3 | IC50 | 2 | — | |
CQEKMSRTDPXHST
|
8.2 | IC50 | 2 | — | |
JYNPEZDAIHSJHW
|
8.2 | IC50 | 2 | — | |
PZJQTRGWISHVPT
|
8.2 | IC50 | 2 | — | |
SBYNVOVSJLOHRE
|
8.2 | IC50 | 2 | — | |
LAHPLBHKJGGIEF
|
8.2 | IC50 | 2 | — | |
MMQLCGFOEBSWCN
|
8.2 | IC50 | 2 | — | |
OWWNUAVAXAAAAM
|
8.2 | IC50 | 2 | — | |
DGPCIFPFGHXRIB
|
8.2 | IC50 | 2 | — |