Target Details
| UniProt AC | Q13131 |
|---|---|
| Gene Symbol | PRKAA1 |
| Protein Name | 5'-AMP-activated protein kinase catalytic subunit alpha-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF16579 (AdenylateSensor) PF21147 (AMPK_alpha_AID) PF00069 (Pkinase) |
Summary
- Multi-target molecules 282
- Clinical molecules 27
- Avg pChEMBL 6.8
KEGG Pathways (20)
- AMPK signaling pathway
- Adipocytokine signaling pathway
- Alcoholic liver disease
- Apelin signaling pathway
- Autophagy - animal
- Circadian rhythm
- Fluid shear stress and atherosclerosis
- FoxO signaling pathway
- Glucagon signaling pathway
- Hypertrophic cardiomyopathy
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- Non-alcoholic fatty liver disease
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Thermogenesis
- Tight junction
- mTOR signaling pathway
Active Molecules (282)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QVNZKVACBBTKSL
|
6.1 | Ki | 38 | — | |
RIBBPSYZBQQTQC
|
6.1 | Ki | 15 | — | |
RVSKJUNTDGBSSS
|
6.1 | Ki | 25 | — | |
UJBJWYNPUOLFIZ
|
6.1 | Ki | 49 | — | |
UXUQVXDYXKMCGA
|
6.1 | Ki | 21 | — | |
UYJNQQDJUOUFQJ
|
6.1 | Ki | 68 | — | |
XPHWIERLJBFPFV
|
6.1 | Ki | 69 | — | |
ZVWRFVCNQOECJS
|
6.1 | Ki | 71 | — | |
UKBGBACORPRCGG
|
6.1 | IC50 | 17 | — | |
ZWIGVNWZHBPXNS
|
6.1 | IC50 | 7 | — | |
HRKJFKJZUNJKNU
|
6.1 | IC50 | 10 | — | |
KGMVZSJAPXYTKH
|
6.1 | IC50 | 23 | — | |
LQVXSNNAFNGRAH
|
6.1 | Kd | 33 | Yes | |
BUMYTKZYNNGHLL
|
6.0 | IC50 | 7 | — | |
WWTRFWLRGARRAD
|
6.0 | IC50 | 10 | — | |
SVJBHQPXESBDEQ
|
6.0 | IC50 | 9 | — | |
FCJGMZMSVIAAJU
|
6.0 | IC50 | 9 | — | |
AHJRHEGDXFFMBM
|
6.0 | Ki | 28 | — | |
GQHMZZXJWGPHDA
|
6.0 | Ki | 20 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
LYNBNVBMAGDJRW
|
6.0 | Ki | 81 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MFMXAWQGPQXDRJ
|
6.0 | Ki | 27 | — | |
OWFLADWRSCINST
|
6.0 | Ki | 30 | — | |
PNKALLUVKOKYHZ
|
6.0 | Ki | 32 | — | |
PSCJSWRVCKUMSL
|
6.0 | Ki | 35 | — | |
SEZFNTZQMWJIAI
|
6.0 | Ki | 22 | — | |
SRUYMJRFVGLQDV
|
6.0 | Ki | 37 | — | |
UQJQNZHGEVLHST
|
6.0 | Ki | 15 | — | |
XYXLUJQBBIBJFV
|
6.0 | Ki | 36 | — | |
ZHRYDDVDLCQYQA
|
6.0 | Ki | 5 | — |