Target Details
| UniProt AC | Q13131 |
|---|---|
| Gene Symbol | PRKAA1 |
| Protein Name | 5'-AMP-activated protein kinase catalytic subunit alpha-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF16579 (AdenylateSensor) PF21147 (AMPK_alpha_AID) PF00069 (Pkinase) |
Summary
- Multi-target molecules 282
- Clinical molecules 27
- Avg pChEMBL 6.8
KEGG Pathways (20)
- AMPK signaling pathway
- Adipocytokine signaling pathway
- Alcoholic liver disease
- Apelin signaling pathway
- Autophagy - animal
- Circadian rhythm
- Fluid shear stress and atherosclerosis
- FoxO signaling pathway
- Glucagon signaling pathway
- Hypertrophic cardiomyopathy
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- Non-alcoholic fatty liver disease
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Thermogenesis
- Tight junction
- mTOR signaling pathway
Active Molecules (282)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MLSDVCJXCYFKAJ
|
6.8 | IC50 | 3 | — | |
NOGWJYQSYBAMTO
|
6.8 | Kd | 3 | — | |
UDMBCSSLTHHNCD
|
6.8 | Kd | 11 | — | |
AUDNGNGLLRZLDR
|
6.8 | Ki | 33 | — | |
DBXGGXLBTWZXBB
|
6.8 | Ki | 39 | — | |
DKZYXHCYPUVGAF
|
6.8 | Kd | 112 | — | |
GJOXRIYWDHESDF
|
6.8 | Ki | 27 | — | |
LBVKEEFIPBQIMD
|
6.8 | Ki | 27 | — | |
LOCWELCIOZHZHE
|
6.8 | Ki | 11 | — | |
SDBOIBYRBWPIEL
|
6.8 | Ki | 31 | — | |
VNDWQCSOSCCWIP
|
6.8 | Ki | 39 | Yes | |
XIOOJUQFJYPVLA
|
6.8 | Ki | 17 | — | |
YEHCNYAQEBQCCS
|
6.8 | Ki | 74 | — | |
YWTBGJGMTBHQTM
|
6.8 | Ki | 65 | — | |
ZGDYBJXDIXVTLV
|
6.8 | Ki | 54 | — | |
PIPKBPQXMOCACO
|
6.8 | IC50 | 2 | — | |
HTVNZZYDHQNFBS
|
6.8 | IC50 | 3 | — | |
BMGQWWVMWDBQGC
|
6.7 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.7 | Kd | 91 | Yes | |
BZYRCHBRDGOULK
|
6.7 | IC50 | 2 | — | |
LIZNIAKSBJKPQC
|
6.7 | IC50 | 3 | — | |
BPNUQXPIQBZCMR
|
6.7 | Ki | 60 | — | |
GUBJNPWVIUFSTR
|
6.7 | Kd | 103 | — | |
GZCJKJJWOUAGMR
|
6.7 | Kd | 3 | — | |
LKUJDAHYLPICSE
|
6.7 | Ki | 24 | — | |
LLRSNVNZYTWKPN
|
6.7 | IC50 | 7 | — | |
NDBJFFCSTXBTFV
|
6.7 | IC50 | 6 | — | |
NKGLJTITEFZKAN
|
6.7 | Ki | 35 | — | |
OEEGUWWPGAZRIJ
|
6.7 | Ki | 21 | — | |
ORQCQXMGDYAIOI
|
6.7 | IC50 | 6 | — | |
OUJZYQBEFNDJQN
|
6.7 | Ki | 71 | — | |
WAKGEHXTOOFEAE
|
6.7 | Ki | 27 | — | |
XSRHBCYNCKAFKS
|
6.7 | Ki | 45 | — | |
ZSSGLTYUJFFIAZ
|
6.7 | IC50 | 2 | — | |
IUDLPZTURGVXEA
|
6.7 | Kd | 7 | — | |
WNDUJGBGBDASMN
|
6.7 | IC50 | 2 | — | |
YJKYSCKYOBZSRV
|
6.7 | Kd | 3 | — | |
CBVYRMZAJKSDGJ
|
6.7 | IC50 | 2 | — | |
HEPDAJRNJBNJAE
|
6.7 | IC50 | 15 | Yes | |
JPQIKBXALJNAKG
|
6.7 | IC50 | 3 | — | |
HCSLNMZYDZLMOP
|
6.6 | IC50 | 3 | — | |
PIVGOZQUWKCUID
|
6.6 | IC50 | 7 | — | |
UJGXTMZILSGDLG
|
6.6 | IC50 | 5 | Yes | |
AWDORCFLUJZUQS
|
6.6 | Ki | 22 | — | |
CKVWQORGCCEYHS
|
6.6 | Ki | 50 | — | |
DPEXRCOBPACFOO
|
6.6 | Ki | 36 | — | |
GHPFSYCYZJKVDZ
|
6.6 | Ki | 18 | Yes | |
HAYYBYPASCDWEQ
|
6.6 | Ki | 47 | — | |
HSKVRPZJBMXFDX
|
6.6 | Ki | 20 | — | |
QPORZABOFXPRHM
|
6.6 | Ki | 18 | — |