Target Details
| UniProt AC | Q13126 |
|---|---|
| Gene Symbol | MTAP |
| Protein Name | S-methyl-5'-thioadenosine phosphorylase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01048 (PNP_UDP_1) |
Summary
- Multi-target molecules 11
- Clinical molecules 0
- Avg pChEMBL 8.8
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (11)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MZZBHZOHYGEGEE
|
11.0 | Kd | 3 | — | |
NTHMDFGHOCNNOE
|
10.1 | Ki | 4 | — | |
FYNHVLXSUCFVCL
|
9.8 | Ki | 3 | — | |
VWBWUCDQZUSUQC
|
9.6 | Ki | 3 | — | |
DIGGNILBPCEZIV
|
9.2 | Ki | 3 | — | |
PLIGEAXYYNDCDB
|
9.0 | Ki | 3 | — | |
PLIGEAXYYNDCDB
|
9.0 | Ki | 2 | — | |
YTSGCQRBVYKQCC
|
8.7 | Ki | 4 | — | |
FMPORPLMRXTYNC
|
7.6 | Kd | 3 | — | |
YYIVMSWPFALBOP
|
6.8 | Ki | 4 | — | |
NTHMDFGHOCNNOE
|
6.1 | Ki | 2 | — |