Target Details
| UniProt AC | Q13043 |
|---|---|
| Gene Symbol | STK4 |
| Protein Name | Serine/threonine-protein kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11629 (Mst1_SARAH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 94
- Clinical molecules 15
- Avg pChEMBL 6.8
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (94)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GCIKSSRWRFVXBI
|
6.7 | Kd | 109 | Yes | |
HUAPVUVLSXALII
|
6.7 | IC50 | 3 | — | |
PIQCTGMSNWUMAF
|
6.7 | Kd | 137 | Yes | |
ZKQLNNVJKSTDGB
|
6.7 | IC50 | 2 | — | |
ZCBUQCWBWNUWSU
|
6.7 | Kd | 59 | — | |
ZWDUUSQSMVRZHV
|
6.7 | IC50 | 3 | — | |
ALKJNCZNEOTEMP
|
6.6 | Kd | 55 | — | |
NMUOPBMRTBMZGB
|
6.6 | IC50 | 2 | — | |
XZKDYHDTDSBKKV
|
6.6 | IC50 | 2 | — | |
UJLAWZDWDVHWOW
|
6.6 | Kd | 4 | — | |
JWNPDZNEKVCWMY
|
6.6 | Kd | 57 | Yes | |
XIVPVCPBGAFXJA
|
6.6 | IC50 | 2 | — | |
YXFNNHJWPFANTQ
|
6.5 | IC50 | 3 | — | |
QQWUGDVOUVUTOY
|
6.5 | Kd | 231 | Yes | |
CVJJGKHSVZTCSY
|
6.3 | IC50 | 2 | — | |
DEUHRYNUMMEYHI
|
6.3 | IC50 | 2 | — | |
DIABFIQALHQONE
|
6.3 | IC50 | 2 | — | |
IBOVLFFYQWKZFN
|
6.3 | IC50 | 2 | — | |
LBWANVYGDFHTRC
|
6.3 | IC50 | 2 | — | |
LZVQWGYDMCTNJC
|
6.3 | IC50 | 2 | — | |
MIURWHKJMYMLCP
|
6.3 | IC50 | 2 | — | |
MPDAGVPGHCHPMC
|
6.3 | IC50 | 2 | — | |
MXEUNJLZLFMHOA
|
6.3 | IC50 | 2 | — | |
NEWMPWSBRISBBJ
|
6.3 | IC50 | 2 | — | |
PDUOASXHLKZWEN
|
6.3 | IC50 | 2 | — | |
PRZMXPRPGHYMHN
|
6.3 | IC50 | 2 | — | |
RIUCXIZLRCRCFO
|
6.3 | IC50 | 2 | — | |
UHKXLPHLKSGYPI
|
6.3 | IC50 | 2 | — | |
VNHDCNPUZFAZKU
|
6.3 | IC50 | 2 | — | |
VWNJEWMXAGIYCW
|
6.3 | IC50 | 2 | — | |
YLYXECAEEDEGIO
|
6.3 | IC50 | 2 | — | |
ZSBOVIKNCKVUHX
|
6.3 | IC50 | 2 | — | |
YYLKKYCXAOBSRM
|
6.2 | Kd | 191 | — | |
KTEIFNKAUNYNJU
|
6.2 | Kd | 114 | — | |
XKFTZKGMDDZMJI
|
6.2 | Kd | 64 | Yes | |
DYNHJHQFHQTFTP
|
6.2 | Kd | 38 | — | |
ZZSBPGIGIUFJRA
|
6.1 | Kd | 46 | — | |
QZZMUIJVVAGHJA
|
6.1 | IC50 | 3 | — | |
RYYNGWLOYLRZLK
|
6.1 | Kd | 45 | — | |
TZWUTAYHWCWNFP
|
6.1 | IC50 | 3 | — | |
PDOQBOJDRPLBQU
|
6.1 | Kd | 21 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |