Target Details
| UniProt AC | Q13043 |
|---|---|
| Gene Symbol | STK4 |
| Protein Name | Serine/threonine-protein kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11629 (Mst1_SARAH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 94
- Clinical molecules 15
- Avg pChEMBL 6.8
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (94)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.7 | Kd | 213 | — | |
HKSZLNNOFSGOKW
|
9.3 | Kd | 408 | — | |
UIARLYUEJFELEN
|
8.5 | Kd | 289 | Yes | |
OSVUGUHRKMMBSE
|
8.4 | Kd | 170 | — | |
NXSJMRCTGYTSTK
|
8.2 | Kd | 200 | — | |
XZXHXSATPCNXJR
|
8.1 | Kd | 165 | Yes | |
WINHZLLDWRZWRT
|
7.7 | Kd | 201 | Yes | |
KOZFSFOOLUUIGY
|
7.5 | Kd | 88 | Yes | |
MWKSRKSEWLRPBL
|
7.4 | Kd | 1075 | — | |
BMGQWWVMWDBQGC
|
7.4 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
7.4 | Kd | 91 | Yes | |
GUBJNPWVIUFSTR
|
7.3 | Kd | 103 | — | |
ONFLVQULIQDDSN
|
7.3 | IC50 | 3 | — | |
IAYGCINLNONXHY
|
7.2 | Kd | 50 | — | |
AYRVYPOFYQSRNH
|
7.2 | IC50 | 2 | — | |
QMQJFRBEIOAQNT
|
7.2 | IC50 | 3 | — | |
DKZYXHCYPUVGAF
|
7.2 | Kd | 112 | — | |
YRDHKIFCGOZTGD
|
7.2 | IC50 | 21 | — | |
FWEIAKDAIDQPRK
|
7.1 | IC50 | 2 | — | |
QGACVLPEELTUQG
|
7.1 | IC50 | 2 | — | |
XRCXPEPDTZGHNO
|
7.0 | IC50 | 2 | — | |
JKHBVOCOHYSWTQ
|
7.0 | IC50 | 3 | — | |
JMAPTHRNJHOVDP
|
7.0 | IC50 | 3 | — | |
NCXSLSJEOUOJBB
|
7.0 | IC50 | 3 | — | |
BLLJUCXNHUVEHL
|
7.0 | IC50 | 3 | — | |
PBCZSGKMGDDXIJ
|
6.9 | Kd | 68 | Yes | |
QHWXURVXTQGCOB
|
6.9 | IC50 | 3 | — | |
QWHANLNIEKAAFF
|
6.9 | IC50 | 2 | — | |
SLOIJUIDHUKLRX
|
6.9 | IC50 | 3 | — | |
VQVBIURGGWKQOR
|
6.9 | IC50 | 2 | — | |
ZWVZORIKUNOTCS
|
6.9 | IC50 | 10 | Yes | |
VCZPJHYQIPIKSV
|
6.9 | IC50 | 3 | — | |
CTNPALGJUAXMMC
|
6.9 | Kd | 151 | — | |
KDKUVYLMPJIGKA
|
6.9 | Kd | 91 | Yes | |
DJOLWWBENMZSKJ
|
6.9 | IC50 | 2 | — | |
OICKVPGRZUWXPB
|
6.9 | IC50 | 3 | — | |
AFBCNAMQWNEPEP
|
6.8 | IC50 | 2 | — | |
HVELYDDHAUZMMJ
|
6.8 | IC50 | 2 | — | |
SJUNPBBKTNPXAO
|
6.8 | IC50 | 2 | — | |
RQJDPSBBHHYXOK
|
6.8 | IC50 | 2 | — | |
SUBYPZBREZXPCW
|
6.8 | IC50 | 3 | — | |
BHTWDJBVZQBRKP
|
6.8 | IC50 | 4 | — | |
QSJSVHCOJILSCM
|
6.8 | IC50 | 2 | — | |
RCRFSYHNZNAAKZ
|
6.8 | IC50 | 2 | — | |
FZMKVQZVEVRANJ
|
6.8 | IC50 | 2 | — | |
AXVWXYOCYXZGCZ
|
6.8 | IC50 | 3 | — | |
FZIPVCYYDYBQOZ
|
6.7 | IC50 | 2 | — | |
MUOUHNBOXJIELS
|
6.7 | IC50 | 3 | — | |
UBPYILGKFZZVDX
|
6.7 | IC50 | 130 | Yes | |
XCAXLCSQKKQKHA
|
6.7 | IC50 | 3 | — |