Target Details
| UniProt AC | Q13003 |
|---|---|
| Gene Symbol | GRIK3 |
| Protein Name | Glutamate receptor ionotropic, kainate 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01094 (ANF_receptor) PF00060 (Lig_chan) PF10613 (Lig_chan-Glu_bd) |
Summary
- Multi-target molecules 16
- Clinical molecules 0
- Avg pChEMBL 6.74
KEGG Pathways (3)
Active Molecules (16)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VZFRNCSOCOPNDB
|
8.3 | Ki | 3 | — | |
VLSMHEGGTFMBBZ
|
8.0 | Ki | 5 | — | |
NHFLJQCBAJUWAE
|
7.4 | Ki | 3 | — | |
ONWXFZVXNOZZFR
|
7.3 | Ki | 9 | — | |
PIWNUFICDRESOQ
|
7.0 | Ki | 9 | — | |
YXQUINDTMKETDY
|
7.0 | Ki | 9 | — | |
MCKOVZZCGOMMIB
|
6.8 | Ki | 6 | — | |
KTYABWSAGQKAPP
|
6.4 | Ki | 9 | — | |
NAVAGRCBXRSPTH
|
6.4 | Ki | 2 | — | |
AYWSXMRAQKWRMH
|
6.3 | Ki | 3 | — | |
DHOYHGUZQYPTFA
|
6.3 | Ki | 2 | — | |
KNAYYBRIBNEIAL
|
6.2 | Ki | 2 | — | |
UWBHJOVXAJRYJM
|
6.2 | Ki | 2 | — | |
WYJNVGSFRNBGEH
|
6.2 | Ki | 9 | — | |
WHUUTDBJXJRKMK
|
6.1 | Ki | 5 | — | |
WHUUTDBJXJRKMK
|
6.1 | Ki | 20 | — |