Target Details
| UniProt AC | Q13002 |
|---|---|
| Gene Symbol | GRIK2 |
| Protein Name | Glutamate receptor ionotropic, kainate 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01094 (ANF_receptor) PF00060 (Lig_chan) PF10613 (Lig_chan-Glu_bd) |
Summary
- Multi-target molecules 19
- Clinical molecules 0
- Avg pChEMBL 6.85
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (19)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YUSZFKPLFIQTGF
|
8.9 | Ki | 2 | — | |
VZFRNCSOCOPNDB
|
8.2 | Ki | 3 | — | |
KRKRAOXTGDJWNI
|
8.0 | Ki | 2 | — | |
VLSMHEGGTFMBBZ
|
7.5 | Ki | 5 | — | |
OXQXJYQSWZFDBB
|
7.3 | Ki | 2 | — | |
NHFLJQCBAJUWAE
|
7.3 | Ki | 3 | — | |
PIWNUFICDRESOQ
|
7.0 | Ki | 9 | — | |
YXQUINDTMKETDY
|
7.0 | Ki | 9 | — | |
LRUYIRXPCIHVCY
|
6.8 | Ki | 2 | — | |
TYAXDMDRDFQFHK
|
6.5 | Ki | 2 | — | |
KTYABWSAGQKAPP
|
6.4 | Ki | 9 | — | |
RCCMXKJGURLWPB
|
6.3 | Ki | 4 | — | |
KXNAWNLNEPJGOW
|
6.3 | Ki | 2 | — | |
MKAFLUPVNVGIOL
|
6.2 | Ki | 2 | — | |
ONWXFZVXNOZZFR
|
6.2 | Ki | 9 | — | |
WYJNVGSFRNBGEH
|
6.2 | Ki | 9 | — | |
LRUYIRXPCIHVCY
|
6.1 | Ki | 2 | — | |
MCKOVZZCGOMMIB
|
6.0 | Ki | 6 | — | |
WJHKVWNKYRFLBD
|
6.0 | Ki | 2 | — |