Target Details
| UniProt AC | Q12884 |
|---|---|
| Gene Symbol | FAP |
| Protein Name | Prolyl endopeptidase FAP |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00930 (DPPIV_N) PF00326 (Peptidase_S9) |
Summary
- Multi-target molecules 366
- Clinical molecules 0
- Avg pChEMBL 8.84
Active Molecules (366)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PVWNTNVPPWCQAH
|
6.2 | IC50 | 2 | — | |
BTGXNIALOLYGDP
|
6.2 | IC50 | 2 | — | |
MEPRZPLBMXAVKQ
|
6.2 | IC50 | 3 | — | |
LHBJCBLEWINWEE
|
6.2 | IC50 | 3 | — | |
OXWKYGRZWVLPOF
|
6.2 | IC50 | 4 | — | |
XGNBIYXILDDDQR
|
6.2 | IC50 | 4 | — | |
XTKKBNBCZVXQHF
|
6.1 | IC50 | 2 | — | |
WDLHHKVPFXMOGF
|
6.1 | Ki | 2 | — | |
ZWKWPVARAOYCNW
|
6.1 | IC50 | 2 | — | |
NMGHEGWLIMQXHB
|
6.1 | IC50 | 3 | — | |
AYKSOEXCVFOICI
|
6.1 | IC50 | 2 | — | |
XJERLNGAISBIJH
|
6.1 | IC50 | 2 | — | |
DYSZJGFBTWPUEV
|
6.0 | Ki | 5 | — | |
MHAGASFEHUMNPA
|
6.0 | IC50 | 2 | — | |
AUZSDJGYAUSLSY
|
6.0 | IC50 | 2 | — | |
BJBOAPYAMPEKGS
|
6.0 | IC50 | 2 | — |