Target Details
| UniProt AC | Q12884 |
|---|---|
| Gene Symbol | FAP |
| Protein Name | Prolyl endopeptidase FAP |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00930 (DPPIV_N) PF00326 (Peptidase_S9) |
Summary
- Multi-target molecules 366
- Clinical molecules 0
- Avg pChEMBL 8.84
Active Molecules (366)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XAUBWUDBHMPSMA
|
7.1 | IC50 | 2 | — | |
IWHLQEBGPICVMJ
|
7.1 | IC50 | 7 | — | |
LTXREWYXXSTFRX
|
7.0 | IC50 | 3 | — | |
HWDDQAHIIBHBMA
|
7.0 | Ki | 2 | — | |
SJCJCRMVAKSLPL
|
7.0 | IC50 | 2 | — | |
BZOKGOVFXOVEJF
|
7.0 | IC50 | 3 | — | |
CXNQIJKSLCMIBD
|
7.0 | IC50 | 2 | — | |
PONJCFYHFPIYJJ
|
7.0 | IC50 | 2 | — | |
SBBQYCLBXQJVIG
|
7.0 | IC50 | 4 | — | |
VRLDMKRCCWBNMD
|
7.0 | IC50 | 2 | — | |
ZEEIEDLWUIHWCQ
|
7.0 | IC50 | 2 | — | |
LKIQQVFCAWXCIN
|
6.9 | IC50 | 2 | — | |
XFMQHPPOMXTIHI
|
6.9 | IC50 | 2 | — | |
MKKPRMVFQDFZMI
|
6.9 | IC50 | 2 | — | |
ZEMFLZQUUHJMGT
|
6.9 | IC50 | 6 | — | |
BJXRITATJHJPJM
|
6.8 | Ki | 2 | — | |
MPZCONICLYEKDC
|
6.8 | IC50 | 3 | — | |
YIYAUIWJPDJXEC
|
6.8 | IC50 | 2 | — | |
GVCXDPXWUCFOOE
|
6.8 | Ki | 3 | — | |
PCRACKRCKRHQQW
|
6.8 | IC50 | 2 | — | |
DGGYQQCWHVPZRV
|
6.8 | IC50 | 3 | — | |
UPJTZJORKZXCFX
|
6.8 | IC50 | 4 | — | |
YZYFOKXDBHHJLB
|
6.8 | IC50 | 5 | — | |
RORVKNCKCFHQRE
|
6.8 | Ki | 2 | — | |
HRRDDUUHRLZHKI
|
6.8 | IC50 | 2 | — | |
PVJXCUHDUBMQIG
|
6.7 | IC50 | 3 | — | |
YSKGDNNCJVHEKT
|
6.7 | Ki | 2 | — | |
LMCNNCISVGRBQK
|
6.7 | IC50 | 3 | — | |
YWWWYGQQSBBBEZ
|
6.6 | Ki | 5 | — | |
FYJNFZCANSKRDW
|
6.6 | Ki | 2 | — | |
FYLALFHFEDXUNH
|
6.6 | IC50 | 3 | — | |
ZRWMIHVRYPKICQ
|
6.6 | IC50 | 2 | — | |
BODWWFCPUUAGKO
|
6.5 | IC50 | 2 | — | |
HFUIIUHINNYZIC
|
6.5 | IC50 | 3 | — | |
CDYUFFXWJNHDCH
|
6.5 | IC50 | 3 | — | |
AHJACGWELFVRGL
|
6.5 | IC50 | 2 | — | |
METFGSCNIQTFJC
|
6.5 | Ki | 2 | — | |
UFKZUCRYERHLMO
|
6.5 | IC50 | 3 | — | |
VEWKBTTWHTZHER
|
6.5 | IC50 | 7 | — | |
KQPQOENOYPKDIN
|
6.4 | IC50 | 2 | — | |
WDWDEKNARRTAAI
|
6.4 | IC50 | 2 | — | |
YPMDOGSZRWVDOZ
|
6.4 | Ki | 6 | — | |
OJFSBKDDVWJMOU
|
6.3 | IC50 | 2 | — | |
SNWSTRLFSXYKCV
|
6.3 | IC50 | 2 | — | |
WWMPHWQJWJIWRD
|
6.3 | IC50 | 3 | — | |
DTSZQBAFUITGDQ
|
6.3 | Ki | 4 | — | |
NEGWJHQAWQAHOF
|
6.3 | Ki | 5 | — | |
AWKXFOWHVYKTSA
|
6.3 | IC50 | 2 | — | |
SWAHNRUQLSQRJA
|
6.3 | IC50 | 3 | — | |
OOTQGBQMGZXPSV
|
6.3 | Ki | 4 | — |