Target Details
| UniProt AC | Q12884 |
|---|---|
| Gene Symbol | FAP |
| Protein Name | Prolyl endopeptidase FAP |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00930 (DPPIV_N) PF00326 (Peptidase_S9) |
Summary
- Multi-target molecules 366
- Clinical molecules 0
- Avg pChEMBL 8.84
Active Molecules (366)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BMCGYCXNUMDZSH
|
7.8 | IC50 | 6 | — | |
LLZDDETUMYCFPV
|
7.7 | IC50 | 2 | — | |
ZAARZJZAJFNJOU
|
7.7 | IC50 | 2 | — | |
ZHPLOOABVYXWII
|
7.7 | IC50 | 2 | — | |
FKCMADOPPWWGNZ
|
7.7 | IC50 | 6 | — | |
IBTPVUMVMUNDFX
|
7.7 | IC50 | 2 | — | |
KXDXUFDMNMEQHZ
|
7.7 | Ki | 2 | — | |
NEYFNISEEPBUIQ
|
7.7 | IC50 | 2 | — | |
RDORJWTZVFNEPH
|
7.7 | IC50 | 2 | — | |
ZETKDIGBGDRCMD
|
7.7 | IC50 | 2 | — | |
WYBXEQQFDLJIFJ
|
7.7 | IC50 | 2 | — | |
NHEGAZXGGOIPDR
|
7.6 | IC50 | 2 | — | |
UUOZISWTWURDGU
|
7.6 | Ki | 3 | — | |
ZWYYINYQGNXKPK
|
7.6 | IC50 | 2 | — | |
IZHXCXLXFBTXRG
|
7.6 | IC50 | 3 | — | |
ZMQPTBIGGCCUBB
|
7.6 | IC50 | 2 | — | |
MQHXRECXBSFFAH
|
7.6 | IC50 | 6 | — | |
DLADMVKMDFATLY
|
7.6 | IC50 | 2 | — | |
NTVCUWWTUPIBEG
|
7.5 | IC50 | 2 | — | |
HWVLQZVEKAYKOF
|
7.5 | Ki | 2 | — | |
XSBZZZGVAIXJLD
|
7.5 | IC50 | 6 | — | |
DRBWRJPFNOBNIO
|
7.5 | IC50 | 2 | — | |
ITLZQNVDXDVBBF
|
7.5 | IC50 | 5 | — | |
SCBANKPTATZMOP
|
7.5 | IC50 | 3 | — | |
VFMUPQNVIIFBNS
|
7.5 | IC50 | 3 | — | |
XBIIDVIXTFCFMM
|
7.5 | IC50 | 5 | — | |
YLQGXGBOYJWXBT
|
7.5 | IC50 | 6 | — | |
SZABTEXPMLELKZ
|
7.5 | IC50 | 2 | — | |
FJQWIWSFPZONQA
|
7.5 | IC50 | 2 | — | |
MZIWWENHLVYLFI
|
7.5 | IC50 | 2 | — | |
ATPDSSDINQDMAK
|
7.4 | IC50 | 2 | — | |
PHCFSFBQEROREL
|
7.4 | IC50 | 6 | — | |
WDFZXMUIFGGBQF
|
7.4 | IC50 | 6 | — | |
PDSFQJYJMMJUTN
|
7.3 | IC50 | 3 | — | |
QWHOCVLSWYFAHP
|
7.3 | IC50 | 2 | — | |
JTKCHMXVNWZDGD
|
7.3 | IC50 | 3 | — | |
DPUGQHXSZXEHQR
|
7.3 | IC50 | 2 | — | |
XGTQGHHNJPRPPY
|
7.3 | Ki | 2 | — | |
BZTBBVKEKPNNBE
|
7.3 | IC50 | 4 | — | |
HGEQTKWTBCNJEW
|
7.3 | IC50 | 4 | — | |
XOHYLGURIBTWKB
|
7.3 | IC50 | 2 | — | |
FWTKUAZIABBHDG
|
7.2 | IC50 | 5 | — | |
DOZHWRXRWJVMNP
|
7.2 | IC50 | 2 | — | |
OXVITDRTBPKXQR
|
7.2 | IC50 | 2 | — | |
DDSNGWWAXQJNCU
|
7.2 | IC50 | 2 | — | |
JVPBPORZRDYLOU
|
7.1 | IC50 | 6 | — | |
SEAKPEIATATKKD
|
7.1 | IC50 | 7 | — | |
ZNNCLYSYFNMXCX
|
7.1 | IC50 | 7 | — | |
GRAXWJMKESEPHA
|
7.1 | IC50 | 2 | — | |
NCKFTUHNPCXRDM
|
7.1 | IC50 | 6 | — |