Target Details
| UniProt AC | Q12884 |
|---|---|
| Gene Symbol | FAP |
| Protein Name | Prolyl endopeptidase FAP |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00930 (DPPIV_N) PF00326 (Peptidase_S9) |
Summary
- Multi-target molecules 366
- Clinical molecules 0
- Avg pChEMBL 8.84
Active Molecules (366)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MBUXPPRHGGRRKJ
|
9.2 | IC50 | 2 | — | |
NEUOTELYJPSZFF
|
9.2 | IC50 | 3 | — | |
VZMSNDLDHMJHAH
|
9.1 | IC50 | 3 | — | |
ZUEXRXMHJQFNSG
|
9.1 | IC50 | 3 | — | |
HXQISXPMFJMCQZ
|
9.0 | IC50 | 2 | — | |
PAAZUJKETHRPFL
|
9.0 | IC50 | 2 | — | |
UHUQCJJQRNMUJJ
|
9.0 | IC50 | 2 | — | |
VUHBLOBXESFZOE
|
9.0 | IC50 | 2 | — | |
STICQYMSICEAOK
|
9.0 | IC50 | 3 | — | |
RTBMMNRHJFIOCP
|
9.0 | IC50 | 2 | — | |
VEFSZHQQQXLTPA
|
9.0 | IC50 | 3 | — | |
FPNJXNKGPWSIAM
|
8.9 | IC50 | 2 | — | |
BLTYWXMDJBDQPE
|
8.8 | IC50 | 2 | — | |
PCDCFSRMQZWMHF
|
8.8 | IC50 | 3 | — | |
PTVMRWQEZPTMFA
|
8.8 | IC50 | 3 | — | |
GSKJKUOZKRGOTN
|
8.8 | IC50 | 2 | — | |
HTTMQAPXSRDVJM
|
8.8 | IC50 | 2 | — | |
QUTRTBDFCYIXBN
|
8.8 | IC50 | 2 | — | |
ZVKAJJHIUZHVQM
|
8.8 | IC50 | 2 | — | |
PCHRROMHSFRTIA
|
8.7 | IC50 | 2 | — | |
UHYVWZMRNGLLCG
|
8.7 | IC50 | 2 | — | |
PUOOCZVRHBHJRS
|
8.6 | IC50 | 2 | — | |
CIWYCGJKMQVNMP
|
8.5 | IC50 | 3 | — | |
LIXQSARDPQLLTH
|
8.5 | IC50 | 2 | — | |
BIACSSXDUXVEGP
|
8.4 | IC50 | 2 | — | |
DMTPQYQQHYOTQM
|
8.4 | IC50 | 6 | — | |
PDSFQJYJMMJUTN
|
8.3 | IC50 | 3 | — | |
NFVMOVDFHPHEHQ
|
8.3 | IC50 | 2 | — | |
REWJLEXLSFEDEB
|
8.3 | IC50 | 2 | — | |
ABDXIQMAFUNGEW
|
8.2 | IC50 | 2 | — | |
MHFTVQPOSPZQHI
|
8.2 | IC50 | 2 | — | |
MTHMMXFBHKGAAI
|
8.2 | IC50 | 4 | — | |
JVPUEBYYUCOOCE
|
8.2 | IC50 | 2 | — | |
QVGIJGPVKMNEPA
|
8.1 | IC50 | 3 | — | |
QFLFLFSVFRSQHH
|
8.1 | IC50 | 3 | — | |
WEULWCVDIGOEBG
|
8.1 | IC50 | 2 | — | |
WYXUOAHCHCVVCT
|
8.1 | IC50 | 2 | — | |
AOCOAPQOYKJKHO
|
8.1 | IC50 | 2 | — | |
KCDMIYYWRZLEKG
|
8.1 | IC50 | 3 | — | |
CXDSYZLZPXATBE
|
8.0 | IC50 | 3 | — | |
WSPHRNDYNWUWIA
|
8.0 | IC50 | 3 | — | |
ASFLZYSLTQLPGZ
|
8.0 | IC50 | 6 | — | |
FKCMADOPPWWGNZ
|
8.0 | IC50 | 3 | — | |
FKCMADOPPWWGNZ
|
8.0 | IC50 | 5 | — | |
MZKOGMKOZUXLIX
|
8.0 | IC50 | 2 | — | |
YEVNJKBZDRFUJQ
|
7.9 | IC50 | 2 | — | |
YFJWJINWDUEJAY
|
7.9 | Ki | 2 | — | |
BDSCRXMWRYZJKF
|
7.8 | Ki | 2 | — | |
MQHXRECXBSFFAH
|
7.8 | IC50 | 6 | — | |
ODGOFEKKXPASHL
|
7.8 | IC50 | 2 | — |