Target Details
| UniProt AC | Q12884 |
|---|---|
| Gene Symbol | FAP |
| Protein Name | Prolyl endopeptidase FAP |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00930 (DPPIV_N) PF00326 (Peptidase_S9) |
Summary
- Multi-target molecules 366
- Clinical molecules 0
- Avg pChEMBL 8.84
Active Molecules (366)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JPTCGWSZMWKBNF
|
9.8 | IC50 | 2 | — | |
XVHXOTBMIIWVFQ
|
9.8 | IC50 | 2 | — | |
DEKKFTKROMHZAE
|
9.8 | IC50 | 2 | — | |
FIOOWVRFCXACGU
|
9.8 | IC50 | 2 | — | |
GCQBMBDBCYNXPT
|
9.8 | IC50 | 2 | — | |
HKXVFSNOGZOHLU
|
9.8 | IC50 | 2 | — | |
VYNMTICGRXHAEX
|
9.8 | IC50 | 2 | — | |
UZMSUYJNBNRGBW
|
9.8 | IC50 | 2 | — | |
JPTCGWSZMWKBNF
|
9.8 | IC50 | 2 | — | |
XHBMQQSFKKFLER
|
9.8 | IC50 | 2 | — | |
NTOIRWWEGTZLGV
|
9.7 | IC50 | 2 | — | |
VOPNNHRJJXXWIG
|
9.7 | IC50 | 2 | — | |
KNJXEQVOFXBFAQ
|
9.7 | IC50 | 2 | — | |
BWVUUKBVZUQABA
|
9.7 | IC50 | 2 | — | |
FFMDEXFQVBUIPE
|
9.7 | IC50 | 2 | — | |
HAEUDXOACFKIBU
|
9.7 | IC50 | 2 | — | |
UGXOMMHKJRFMMM
|
9.7 | IC50 | 2 | — | |
XQOXYCGIRRYPIG
|
9.7 | IC50 | 2 | — | |
YGOKMUFNHQXIEE
|
9.7 | IC50 | 2 | — | |
RKKYAODNIKZROJ
|
9.7 | IC50 | 2 | — | |
BHQNCMQPFNXCHZ
|
9.7 | IC50 | 2 | — | |
IBTFNORVBDUDPP
|
9.7 | IC50 | 2 | — | |
OGYSFSGIEZNUAX
|
9.7 | IC50 | 2 | — | |
NPVRFLOBVJCIAZ
|
9.7 | IC50 | 2 | — | |
XFZZDFKSDXKGLS
|
9.7 | IC50 | 2 | — | |
USRJWFNTEMWYAC
|
9.6 | IC50 | 2 | — | |
OSTZTECCWMVMOJ
|
9.6 | IC50 | 2 | — | |
MJCMOPDWPSGGTH
|
9.6 | IC50 | 2 | — | |
VUMCZFAMVXKLDC
|
9.6 | IC50 | 2 | — | |
ZDDFAXABYJEGIB
|
9.6 | IC50 | 2 | — | |
NVTSVVCOBJKHKI
|
9.6 | IC50 | 2 | — | |
OLRXKVXITDQZDJ
|
9.6 | IC50 | 2 | — | |
PZLKPRVECOGMLC
|
9.6 | IC50 | 2 | — | |
GPYWLBWBTDOUOC
|
9.5 | IC50 | 2 | — | |
JIGUYYXQAKEPKB
|
9.5 | IC50 | 2 | — | |
KJBZPMGWIYEGPF
|
9.5 | IC50 | 2 | — | |
WUOIRTMHLVMFMN
|
9.5 | IC50 | 2 | — | |
QZYAHNXLJPNYIP
|
9.5 | IC50 | 2 | — | |
HZJGLUIJMJYGMO
|
9.5 | IC50 | 2 | — | |
DUDRYQVTKPGWCP
|
9.4 | IC50 | 3 | — | |
NYJCGFBNRXRVEK
|
9.4 | IC50 | 2 | — | |
ICWDAESAANBIGG
|
9.4 | IC50 | 2 | — | |
RALYIZJPDYRDBD
|
9.4 | IC50 | 3 | — | |
XXBLYSCVXGFMPP
|
9.4 | IC50 | 2 | — | |
OUMOKPXHKUZPLS
|
9.4 | IC50 | 2 | — | |
QHKSBUQBSZTVML
|
9.4 | IC50 | 2 | — | |
NFLFYUMFQNNIPE
|
9.3 | IC50 | 3 | — | |
IZABYRMMVXWDIM
|
9.3 | IC50 | 2 | — | |
NNRPSTLTRISCSQ
|
9.3 | IC50 | 2 | — | |
YBVFBNZKQHCYDQ
|
9.3 | IC50 | 2 | — |