Target Details
| UniProt AC | Q12884 |
|---|---|
| Gene Symbol | FAP |
| Protein Name | Prolyl endopeptidase FAP |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00930 (DPPIV_N) PF00326 (Peptidase_S9) |
Summary
- Multi-target molecules 366
- Clinical molecules 0
- Avg pChEMBL 8.84
Active Molecules (366)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KSOBLFKTCLHCSM
|
10.1 | IC50 | 2 | — | |
MXKCUEGHKAELQK
|
10.1 | IC50 | 2 | — | |
VDZWDPQTNDPQPO
|
10.1 | IC50 | 2 | — | |
CHKVYCQSHMXNCK
|
10.0 | IC50 | 2 | — | |
USORGFOLKXPIBW
|
10.0 | IC50 | 2 | — | |
WTYGDPFXBIYRFB
|
10.0 | IC50 | 2 | — | |
CFLDQRFVNWJHFE
|
10.0 | IC50 | 2 | — | |
UTCUYPONNGGJOS
|
10.0 | IC50 | 2 | — | |
CRXCLUHUPYCNMK
|
10.0 | IC50 | 2 | — | |
BJLGLUYPNLVLIF
|
10.0 | IC50 | 2 | — | |
DLQVNTHAYGOAKV
|
10.0 | IC50 | 2 | — | |
GUVSWENHSYFOQO
|
10.0 | IC50 | 2 | — | |
NAUIGRGGFQAIPT
|
10.0 | IC50 | 2 | — | |
SZDICRGIABOEDK
|
10.0 | IC50 | 2 | — | |
UZMSUYJNBNRGBW
|
10.0 | IC50 | 2 | — | |
IFPDOIWCKGVNKE
|
10.0 | IC50 | 2 | — | |
GCQBMBDBCYNXPT
|
10.0 | IC50 | 2 | — | |
DEAODSSVHZTRGK
|
10.0 | IC50 | 2 | — | |
FGEPCVDFVCNUJI
|
10.0 | IC50 | 2 | — | |
GZVBIFATCRQOFF
|
10.0 | IC50 | 2 | — | |
MXKCUEGHKAELQK
|
10.0 | IC50 | 2 | — | |
MXVMKRSOGUFLRC
|
10.0 | IC50 | 2 | — | |
ONVMYIXRFOPLQH
|
10.0 | IC50 | 2 | — | |
PRFUGRYYLWOJNY
|
10.0 | IC50 | 2 | — | |
QVCNSUHMQLXLRO
|
10.0 | IC50 | 2 | — | |
SPZWXOWEXKQOAD
|
10.0 | IC50 | 2 | — | |
VFBKQWJZWWMGCL
|
10.0 | IC50 | 2 | — | |
VNDCCIPQPPXLQP
|
10.0 | IC50 | 2 | — | |
BORCWPKUTLZLEJ
|
9.9 | IC50 | 2 | — | |
DBXQLWJBJCSPIQ
|
9.9 | IC50 | 2 | — | |
GXDZWHPHISQRGL
|
9.9 | IC50 | 2 | — | |
MVLSIGMPPPBZDC
|
9.9 | IC50 | 2 | — | |
MZNFNQRHDURQTB
|
9.9 | IC50 | 2 | — | |
SDQQEJFBJPMSIH
|
9.9 | IC50 | 2 | — | |
USYUIYMUAPRCLB
|
9.9 | IC50 | 2 | — | |
XDSJWOOECLXJRL
|
9.9 | IC50 | 2 | — | |
ZIOIZQJLKHPESI
|
9.9 | IC50 | 2 | — | |
JDJWNGMVZJPNSD
|
9.9 | IC50 | 2 | — | |
CKVGDSOARKWCHY
|
9.9 | IC50 | 2 | — | |
OTGWSROANXIBHL
|
9.9 | IC50 | 3 | — | |
STIFZLVYZUJQIQ
|
9.9 | IC50 | 2 | — | |
YWOQNTUKYYMGKL
|
9.9 | IC50 | 2 | — | |
CPOVUTLGSGKXBM
|
9.9 | IC50 | 2 | — | |
BPXBTZXUHLCLRG
|
9.9 | IC50 | 2 | — | |
VJOTXRKAYMZPSU
|
9.9 | IC50 | 2 | — | |
GDHMLUIBKBKWQQ
|
9.9 | IC50 | 2 | — | |
MFUXFECMAUFOFT
|
9.9 | IC50 | 2 | — | |
AGKIVRWBXRHEHK
|
9.8 | IC50 | 2 | — | |
VDZWDPQTNDPQPO
|
9.8 | IC50 | 2 | — | |
VJZHWKYEFZNGRM
|
9.8 | IC50 | 2 | — |