Target Details
| UniProt AC | Q12884 |
|---|---|
| Gene Symbol | FAP |
| Protein Name | Prolyl endopeptidase FAP |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00930 (DPPIV_N) PF00326 (Peptidase_S9) |
Summary
- Multi-target molecules 366
- Clinical molecules 0
- Avg pChEMBL 8.84
Active Molecules (366)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MZSJPHANWIKYSE
|
10.3 | IC50 | 2 | — | |
XBGZVMYGSPCXFX
|
10.3 | IC50 | 2 | — | |
INTDZVGJKRMKMW
|
10.2 | IC50 | 2 | — | |
OOAQKKMGVAFCBM
|
10.2 | IC50 | 2 | — | |
VVKJNDDMBVHOAO
|
10.2 | IC50 | 2 | — | |
RRQLPFRONBZMCQ
|
10.2 | Kd | 2 | — | |
YBBXYEGJBAEOFI
|
10.2 | IC50 | 2 | — | |
IYUGSEFCZXOZSD
|
10.2 | IC50 | 3 | — | |
JWGAOFWRRCISDL
|
10.2 | IC50 | 2 | — | |
XTTQCXHOQKGXSN
|
10.2 | IC50 | 2 | — | |
IXWDHXCXBXIWMZ
|
10.2 | IC50 | 2 | — | |
MZNFNQRHDURQTB
|
10.2 | IC50 | 2 | — | |
WOLDVHLVKAURLX
|
10.2 | IC50 | 2 | — | |
DTOQUOQVYYOIJK
|
10.2 | IC50 | 2 | — | |
GMHFYPCAAPSRRZ
|
10.2 | IC50 | 2 | — | |
WIBKMQMPJVPXNY
|
10.2 | IC50 | 2 | — | |
XEMYMAPKYPNBCI
|
10.2 | IC50 | 2 | — | |
BSMDTUXAEWXGBM
|
10.2 | IC50 | 2 | — | |
OCWZFRBGMDVTLA
|
10.2 | IC50 | 2 | — | |
VLJUHLKSEMHETM
|
10.2 | IC50 | 2 | — | |
FWIULPJALJLLTE
|
10.2 | IC50 | 2 | — | |
MVLSIGMPPPBZDC
|
10.2 | IC50 | 2 | — | |
ZRIUEQVZJVHYQY
|
10.2 | IC50 | 2 | — | |
GQSQVUPYGFXZJL
|
10.2 | IC50 | 2 | — | |
LAPUWIJZAPNJMC
|
10.2 | IC50 | 2 | — | |
SGVAQIKNLVFPLW
|
10.2 | IC50 | 2 | — | |
YXBOJNLQVIBFOO
|
10.2 | IC50 | 2 | — | |
ITPHLAQPYZIOAB
|
10.2 | IC50 | 2 | — | |
KZSSCUNWLMOEOQ
|
10.2 | IC50 | 2 | — | |
WIOIJTLTZTWPPU
|
10.2 | IC50 | 2 | — | |
BUQHVWNTBCFZLQ
|
10.1 | IC50 | 2 | — | |
NZTBFSSPSNZERA
|
10.1 | IC50 | 2 | — | |
USORGFOLKXPIBW
|
10.1 | IC50 | 2 | — | |
DGQDJAFQIAPENQ
|
10.1 | IC50 | 2 | — | |
INTDZVGJKRMKMW
|
10.1 | IC50 | 2 | — | |
ZCUROAQBTGFWAZ
|
10.1 | IC50 | 2 | — | |
KVECVNJYBFEXQD
|
10.1 | IC50 | 2 | — | |
XVEGXEQMFNPPDB
|
10.1 | IC50 | 2 | — | |
GRALGYJBJWPSTK
|
10.1 | IC50 | 2 | — | |
HORMWUNSPSWHJB
|
10.1 | IC50 | 2 | — | |
JEJQVXPRRBVAQH
|
10.1 | IC50 | 2 | — | |
OWLCAJFTAXWBIJ
|
10.1 | IC50 | 2 | — | |
WIOIJTLTZTWPPU
|
10.1 | IC50 | 2 | — | |
HIEZCODBJOKGHX
|
10.1 | IC50 | 2 | — | |
HOBKRRYAOBAOEG
|
10.1 | IC50 | 2 | — | |
JSFKORGBLHWIAN
|
10.1 | IC50 | 2 | — | |
KWGYHUJGVSKJKM
|
10.1 | IC50 | 2 | — | |
IXWDHXCXBXIWMZ
|
10.1 | IC50 | 2 | — | |
IYOGJVGDNMBQCE
|
10.1 | IC50 | 2 | — | |
ZIGWYACUKUILOS
|
10.1 | IC50 | 2 | — |