Target Details
| UniProt AC | Q12884 |
|---|---|
| Gene Symbol | FAP |
| Protein Name | Prolyl endopeptidase FAP |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00930 (DPPIV_N) PF00326 (Peptidase_S9) |
Summary
- Multi-target molecules 366
- Clinical molecules 0
- Avg pChEMBL 8.84
Active Molecules (366)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PHTNQLKUKIPWAJ
|
10.8 | IC50 | 2 | — | |
WIBKMQMPJVPXNY
|
10.8 | IC50 | 2 | — | |
UFEHGSNMRSIMAK
|
10.7 | IC50 | 2 | — | |
CMYCEAMZAPXCMW
|
10.6 | IC50 | 2 | — | |
GXOHVKCQCIIEOJ
|
10.6 | IC50 | 2 | — | |
PDZAYTNWXFHGDD
|
10.6 | IC50 | 2 | — | |
UKNCPEXKVPRTFL
|
10.6 | IC50 | 2 | — | |
FJCWDJCPHJIIIU
|
10.6 | IC50 | 2 | — | |
FBSNDOFIQIAZNL
|
10.5 | IC50 | 2 | — | |
YBBXYEGJBAEOFI
|
10.5 | IC50 | 2 | — | |
PZQALERHWWQNQV
|
10.5 | IC50 | 2 | — | |
RJCKCWBOMKVXBE
|
10.5 | IC50 | 2 | — | |
OIUCCXSHLWPFSH
|
10.5 | IC50 | 2 | — | |
MSGBYFPTKFQODA
|
10.5 | IC50 | 3 | — | |
DZFDLHBZEQZMDQ
|
10.5 | IC50 | 2 | — | |
YEQGPQSFILIYSG
|
10.5 | IC50 | 2 | — | |
ARZVSKDNGYNMKF
|
10.4 | IC50 | 2 | — | |
UGMQHBJFZIUCFJ
|
10.4 | IC50 | 2 | — | |
YMKPBGRJCLDCIO
|
10.4 | IC50 | 2 | — | |
KVYKFPIRLGSOEV
|
10.4 | IC50 | 2 | — | |
WMWFELYLXJTGLE
|
10.4 | IC50 | 2 | — | |
WIOIJTLTZTWPPU
|
10.4 | IC50 | 2 | — | |
KOFMZONJMIPXFD
|
10.4 | IC50 | 2 | — | |
NSVGKQYLTLZGPJ
|
10.4 | IC50 | 2 | — | |
CZYBGSCBSVMAID
|
10.4 | IC50 | 2 | — | |
UBGODDCOMDEPAG
|
10.4 | IC50 | 2 | — | |
ZPEJVXVQESRFNL
|
10.4 | IC50 | 2 | — | |
CWHFTQYQWMACLS
|
10.4 | IC50 | 2 | — | |
JDJCBZCRKKUWPF
|
10.4 | IC50 | 2 | — | |
HFBNXJXQQMEDQV
|
10.4 | IC50 | 2 | — | |
RRQLPFRONBZMCQ
|
10.4 | IC50 | 2 | — | |
YEQGPQSFILIYSG
|
10.4 | IC50 | 2 | — | |
BSMDTUXAEWXGBM
|
10.3 | IC50 | 2 | — | |
OUAXIVOQNIIUFY
|
10.3 | IC50 | 2 | — | |
WDJZHXQRJOBNAQ
|
10.3 | IC50 | 2 | — | |
YDYQSOBOSIZNSK
|
10.3 | IC50 | 2 | — | |
ZUVIZSBXPFZZHO
|
10.3 | IC50 | 2 | — | |
QCYFCKJWFGHJHH
|
10.3 | IC50 | 2 | — | |
QMJNQRYLOCIWLK
|
10.3 | IC50 | 2 | — | |
IMSHZPRJWGDNAY
|
10.3 | IC50 | 2 | — | |
JXXCGJFWIFDRIY
|
10.3 | IC50 | 2 | — | |
RIQHVEFFFMJOSS
|
10.3 | IC50 | 2 | — | |
RRKLRQFVYOADOY
|
10.3 | IC50 | 2 | — | |
SOVGHANOYJMEML
|
10.3 | IC50 | 2 | — | |
CRMJTVCWBOMJGG
|
10.3 | IC50 | 2 | — | |
DBVPXLLXZQIPDZ
|
10.3 | IC50 | 2 | — | |
IOYKLDJPKHRJEK
|
10.3 | IC50 | 2 | — | |
JXVFJORPICYGPP
|
10.3 | IC50 | 2 | — | |
CRWCYVOHVXAEMF
|
10.3 | IC50 | 3 | — | |
GBMZYOIEUKCVSL
|
10.3 | IC50 | 2 | — |