Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HPRJYEVMXGJJCS
|
8.1 | IC50 | 4 | — | |
NXSAPRAOMACXRV
|
8.1 | IC50 | 4 | — | |
RADSRRYRWZKEEW
|
8.1 | IC50 | 4 | — | |
RVQLPUNPSVMPIU
|
8.1 | IC50 | 2 | — | |
SYMFPMGEVCPXSZ
|
8.1 | IC50 | 5 | — | |
ZFBBKOBKYNRTOS
|
8.1 | IC50 | 4 | — | |
AMOJZZNHYLYYBD
|
8.1 | IC50 | 2 | — | |
CXDXWPGEWIRDBS
|
8.1 | IC50 | 3 | — | |
CXDXWPGEWIRDBS
|
8.1 | IC50 | 4 | — | |
NRDNLCCXBFBMSJ
|
8.1 | IC50 | 4 | — | |
AWOJPBWFDKHWTR
|
8.1 | IC50 | 2 | — | |
NSLJACGCOKVYOC
|
8.1 | IC50 | 4 | — | |
OUNWKMVWDHVXRC
|
8.1 | IC50 | 2 | — | |
UBJLGYQQFARAFL
|
8.1 | IC50 | 2 | — | |
WIFXWIHQARKSIL
|
8.1 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
8.1 | Kd | 165 | Yes | |
FOSRCRDKVZHMBZ
|
8.1 | IC50 | 4 | — | |
LAPPKEKKVUXSCR
|
8.1 | IC50 | 2 | — | |
LNBTVVMNWXKTFO
|
8.1 | IC50 | 2 | — | |
MQQQNGBBTVKGQZ
|
8.1 | IC50 | 4 | — | |
VPQQWBCSZPCKLB
|
8.1 | IC50 | 4 | — | |
LHGBMCHXJSBVDX
|
8.1 | IC50 | 2 | — | |
MBJBZECMDXNZSX
|
8.1 | IC50 | 2 | — | |
OAIGXMDORWMZJX
|
8.1 | IC50 | 4 | — | |
PFBFUNWWEQQNQB
|
8.1 | IC50 | 4 | — | |
UENPHVZMJZONSS
|
8.1 | IC50 | 4 | — | |
ZSOMRVGPVJNHFO
|
8.1 | IC50 | 3 | — | |
AWWTWYGZSSQDDV
|
8.0 | IC50 | 4 | — | |
CZKFYGCROLKVDT
|
8.0 | IC50 | 3 | — | |
KYIVMAWNIPIMAX
|
8.0 | IC50 | 2 | — | |
OOZMTBCGVZLMGL
|
8.0 | IC50 | 2 | — | |
UMCOITRXYYLVMB
|
8.0 | IC50 | 4 | — | |
FQGZERIFFBAKQS
|
8.0 | IC50 | 4 | — | |
WCQNXVPJWXAGFY
|
8.0 | IC50 | 4 | — | |
DTHWSLYDAOOPOE
|
8.0 | IC50 | 4 | — | |
IGOHZEZLKPSIDE
|
8.0 | IC50 | 4 | — | |
RVMVPBZDKHOVRJ
|
8.0 | IC50 | 4 | — | |
UFXPAIWAISVBLY
|
8.0 | IC50 | 4 | — | |
WTBRDNQZOOILBP
|
8.0 | IC50 | 4 | — | |
ZVKWOODYBNGMEY
|
8.0 | IC50 | 4 | — | |
NUWXKTZRKDGSGW
|
8.0 | IC50 | 2 | — | |
VVTZTRAFXXRFHV
|
8.0 | IC50 | 4 | — | |
WHMMKPWGWNYYFE
|
8.0 | IC50 | 2 | — | |
DSSNAGYVGTYAGH
|
8.0 | IC50 | 10 | — | |
PVPLEDXJDAJQPM
|
8.0 | IC50 | 2 | — | |
WPSAGYVBZPKGAO
|
8.0 | IC50 | 2 | — | |
ZISLJLXCLUQNKA
|
8.0 | IC50 | 3 | — | |
UTBNTDYEJRQXQB
|
8.0 | IC50 | 2 | — | |
DJSUVZWWNNNEDR
|
8.0 | IC50 | 2 | — | |
FWSIMUXTYLCNLB
|
8.0 | IC50 | 2 | — |