Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UVXCGYVEUGYYNC
|
8.2 | IC50 | 3 | — | |
NCGOROUZONSZHC
|
8.2 | IC50 | 2 | — | |
UOUHQYNDRQLKBR
|
8.2 | IC50 | 2 | — | |
XLBBUKKTLCFJHL
|
8.2 | IC50 | 4 | — | |
CUEIYXNRRXDHDN
|
8.2 | IC50 | 4 | — | |
DPXCMTQMIGMPBI
|
8.2 | IC50 | 2 | — | |
FJWZASZEWLWFRB
|
8.2 | IC50 | 3 | — | |
FJWZASZEWLWFRB
|
8.2 | IC50 | 4 | — | |
KNGNXLHOEYCPCZ
|
8.2 | IC50 | 4 | — | |
XBHCTLDKTVHKKG
|
8.2 | IC50 | 3 | — | |
BGFQHBDQBASGDN
|
8.2 | IC50 | 4 | — | |
BTBWDZHSUOGEGB
|
8.2 | IC50 | 3 | — | |
HQGIJNUYLNDDFY
|
8.2 | IC50 | 3 | — | |
BXOIQQLQRZDRGP
|
8.2 | IC50 | 4 | — | |
ROHJEIACUNTGFP
|
8.2 | IC50 | 16 | — | |
CGDYJOFBSKXMDN
|
8.1 | IC50 | 4 | — | |
JMWVQYVMGWIDOO
|
8.1 | IC50 | 3 | — | |
KDBWIIMYOYEZDH
|
8.1 | IC50 | 4 | — | |
NBBXQZAASIMPFD
|
8.1 | IC50 | 4 | — | |
SBQMDXILYZEQDX
|
8.1 | IC50 | 3 | — | |
UDRSARITYRCUFL
|
8.1 | IC50 | 4 | — | |
YYTVUKVXIKXZNG
|
8.1 | IC50 | 4 | — | |
LJTFVODOMNCPCP
|
8.1 | IC50 | 4 | — | |
WFAOCMRUJDNSOA
|
8.1 | IC50 | 2 | — | |
AHZDWGRDNJBCPX
|
8.1 | IC50 | 4 | — | |
CDLLABUAFGKJDH
|
8.1 | IC50 | 2 | — | |
CPNQAVXQGZKRMM
|
8.1 | IC50 | 4 | — | |
DRFSMWIGPWLYCE
|
8.1 | IC50 | 2 | — | |
FHZJANCSCXSLSI
|
8.1 | IC50 | 2 | — | |
GPNOEUDRIWKLGC
|
8.1 | IC50 | 2 | — | |
KQVZUBPWFJXMKN
|
8.1 | IC50 | 3 | — | |
LLGTZIXASKDKRV
|
8.1 | IC50 | 2 | — | |
NRSFBLRHWDDEHB
|
8.1 | IC50 | 4 | — | |
PYIGYDCLFZWCRO
|
8.1 | IC50 | 2 | — | |
SSNOOYVRHMFBIF
|
8.1 | IC50 | 2 | — | |
SVQLYPNPTZVLCF
|
8.1 | IC50 | 2 | — | |
UDIUHDBYJMAEKG
|
8.1 | IC50 | 2 | — | |
UKJAACLEQSSYIE
|
8.1 | IC50 | 2 | — | |
WRADGJQBDXJRIT
|
8.1 | IC50 | 2 | — | |
WVXNSAVVKYZVOE
|
8.1 | IC50 | 92 | — | |
ZMODBJGIKIUPSW
|
8.1 | IC50 | 2 | — | |
BPFIPYIIVJLOML
|
8.1 | IC50 | 3 | — | |
MZDSZIKAVUIXKJ
|
8.1 | IC50 | 3 | — | |
XBEJAJFQAGYRNU
|
8.1 | IC50 | 3 | — | |
IABXKANEKUUGPC
|
8.1 | IC50 | 4 | — | |
JVFSAMBNAXDBQY
|
8.1 | IC50 | 2 | — | |
RNOGFYURWHXLGG
|
8.1 | IC50 | 3 | — | |
SDWTWVXMBPUQSC
|
8.1 | IC50 | 4 | — | |
UGAWJRIPKFUXGB
|
8.1 | IC50 | 2 | — | |
GPXJRVLKUZJOES
|
8.1 | IC50 | 3 | — |