Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SCPFYDCGZSWLOY
|
8.3 | IC50 | 4 | — | |
WEIHLBMGCSGIDR
|
8.3 | IC50 | 4 | — | |
XJVMKCJCQDTBQW
|
8.3 | IC50 | 4 | — | |
DYDGFQGBJUDGKC
|
8.3 | IC50 | 4 | — | |
GKTJDVXAUIHAML
|
8.3 | IC50 | 4 | — | |
GNKRUXYNYRQFDL
|
8.3 | IC50 | 4 | — | |
HMFLIEILARDTTE
|
8.3 | IC50 | 2 | — | |
LHVQWBCPTBYJSL
|
8.3 | IC50 | 4 | — | |
MQTNFIVWBJDJRH
|
8.3 | IC50 | 2 | — | |
PCELUAJFVVOBSI
|
8.3 | IC50 | 4 | — | |
PHINIAPYUBKDAN
|
8.3 | IC50 | 4 | — | |
RWENGGARDXLTTR
|
8.3 | IC50 | 3 | — | |
WPRJOLMYEVNSEK
|
8.3 | IC50 | 2 | — | |
XURDGFSSCIUCAC
|
8.3 | IC50 | 4 | — | |
GKMWSAWIKNLTDH
|
8.3 | IC50 | 4 | — | |
XUZJQPLUDYDVEN
|
8.3 | IC50 | 2 | — | |
CQFHCAGCNILQLR
|
8.3 | IC50 | 3 | — | |
CQFHCAGCNILQLR
|
8.3 | IC50 | 3 | — | |
DLKUKWUHCCFYTF
|
8.3 | IC50 | 3 | — | |
MUSDSMKVOIDEMF
|
8.3 | IC50 | 4 | — | |
VBQLIIKEYZCPOL
|
8.3 | IC50 | 4 | — | |
WDFZKMQYTGAITH
|
8.3 | IC50 | 4 | — | |
XSTKLDSKDZEFSN
|
8.3 | IC50 | 4 | — | |
YKWQGXNPYZYKQY
|
8.3 | IC50 | 4 | — | |
YTOQTXOTRNNBQW
|
8.3 | IC50 | 4 | — | |
ZFBBKOBKYNRTOS
|
8.3 | IC50 | 4 | — | |
BPFIPYIIVJLOML
|
8.3 | IC50 | 4 | — | |
QIJNQRCCSXIKCW
|
8.3 | IC50 | 2 | — | |
UEQGBUCCFMIQCV
|
8.3 | IC50 | 4 | — | |
BOHSEWFNQJXFAO
|
8.3 | IC50 | 4 | — | |
NQSLOMAYSOUYFR
|
8.2 | IC50 | 3 | — | |
ORJFNGOUYHBFPE
|
8.2 | IC50 | 4 | — | |
UZXNBLXFPDDYST
|
8.2 | IC50 | 2 | — | |
VINFIBQGNVEOHD
|
8.2 | IC50 | 4 | — | |
JHLDSSUQVZCRDO
|
8.2 | IC50 | 3 | — | |
JNVWCHOWNOCLHA
|
8.2 | IC50 | 4 | — | |
LLDHGYBXXLQDJD
|
8.2 | IC50 | 2 | — | |
ZBBLIQHYOFPIKP
|
8.2 | IC50 | 4 | — | |
MOIKWCOSENYJDE
|
8.2 | IC50 | 4 | — | |
MRKQEMFQARHIQR
|
8.2 | IC50 | 2 | — | |
HMDDJHHCPSISTL
|
8.2 | IC50 | 4 | — | |
MLEGYBAUGFHNOW
|
8.2 | IC50 | 3 | — | |
RGFGVLQJEABYNU
|
8.2 | IC50 | 3 | — | |
DKAWAHOTJBIOOP
|
8.2 | IC50 | 3 | — | |
HTOALBYXWRQRAR
|
8.2 | IC50 | 3 | — | |
IPOSOQDPXNYXKP
|
8.2 | IC50 | 4 | — | |
JVAUXOQNQAAUBJ
|
8.2 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
8.2 | IC50 | 408 | — | |
HKSZLNNOFSGOKW
|
8.2 | Kd | 213 | — | |
ILTIHYQRKNBZLR
|
8.2 | IC50 | 4 | — |