Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JJXRAZVLEQHSOL
|
8.4 | IC50 | 4 | — | |
JLSYAJGCSIAVIW
|
8.4 | IC50 | 4 | — | |
OEZCGAGJZUCOEB
|
8.4 | IC50 | 2 | — | |
SJBXHRBUEGPULP
|
8.4 | IC50 | 4 | — | |
SMIXLVLRWCBPBA
|
8.4 | IC50 | 4 | — | |
WBDRTUBXAWFAOJ
|
8.4 | IC50 | 4 | — | |
XFDWKMREXUNRTL
|
8.4 | IC50 | 2 | — | |
DKLRVMHGCQHXBG
|
8.4 | IC50 | 4 | — | |
GFIIPWSSHMVXHK
|
8.4 | IC50 | 4 | — | |
HTZHPXKKPOLGTR
|
8.4 | IC50 | 9 | — | |
XZWGQOPSCIYJJG
|
8.4 | IC50 | 2 | — | |
ZTXJBHFBIBXQAC
|
8.4 | IC50 | 4 | — | |
KSIYRLNWOATMQX
|
8.4 | IC50 | 3 | — | |
NPVXOWLPOFYACO
|
8.4 | IC50 | 5 | — | |
PGXKVCTXUZHTHO
|
8.4 | IC50 | 4 | — | |
QFMYLXWZJAXERY
|
8.4 | IC50 | 4 | — | |
SPTBDWLBLZVHRD
|
8.4 | IC50 | 2 | — | |
WNIAHFXCAWIXLI
|
8.4 | IC50 | 2 | — | |
XWOQSDCGEZJRNK
|
8.4 | IC50 | 4 | — | |
ACJPYAYXMSVFMW
|
8.4 | IC50 | 2 | — | |
APPUYFNVFFWYFM
|
8.4 | IC50 | 4 | — | |
GBYPCTVFSGFCSE
|
8.4 | IC50 | 3 | — | |
HQDFMNJNVUENSH
|
8.4 | IC50 | 2 | — | |
MQKBHIPASUSQRC
|
8.4 | IC50 | 3 | — | |
ONIHBIZGUJZDHG
|
8.4 | IC50 | 4 | — | |
UMBIRSZUCJNBHB
|
8.4 | IC50 | 18 | — | |
USGGKJZAODNEBP
|
8.4 | IC50 | 2 | — | |
AGYRCBTVZCTMOP
|
8.3 | IC50 | 4 | — | |
AGYRCBTVZCTMOP
|
8.3 | IC50 | 3 | — | |
BVGJNPJMZYLNBE
|
8.3 | IC50 | 3 | — | |
ITIWLFFFNMDGFN
|
8.3 | IC50 | 4 | — | |
LMEIQSASKHJFEN
|
8.3 | IC50 | 4 | — | |
RATPJUQSJPMXQH
|
8.3 | IC50 | 4 | — | |
VIPDXSZEKZMOAC
|
8.3 | IC50 | 3 | — | |
BZUTZGPXMWEYRV
|
8.3 | IC50 | 3 | — | |
DEOQMORRIDRHPD
|
8.3 | IC50 | 3 | — | |
ICAQVATUJCMIBT
|
8.3 | IC50 | 4 | — | |
OASIGFOZMTYWOR
|
8.3 | IC50 | 4 | — | |
SGTSFIPSFBYYSH
|
8.3 | IC50 | 4 | — | |
SJHRIMACUGYDED
|
8.3 | IC50 | 4 | — | |
VWSHIOYTEVXOAS
|
8.3 | IC50 | 4 | — | |
WIXFZICRDRQMNT
|
8.3 | IC50 | 4 | — | |
OOSNHFXEEYPEGT
|
8.3 | IC50 | 3 | — | |
BKANXYVDKHTWQK
|
8.3 | IC50 | 4 | — | |
HQVPUZZSOUVIPN
|
8.3 | IC50 | 4 | — | |
PSPNRRHQXRHIMO
|
8.3 | IC50 | 4 | — | |
CGBNPMZFTROLIN
|
8.3 | IC50 | 4 | — | |
FBBJSCGMJHFVOD
|
8.3 | IC50 | 3 | — | |
QGVUAUSZGWKGSS
|
8.3 | IC50 | 4 | — | |
RIFZMWFVFITGGN
|
8.3 | IC50 | 3 | — |