Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SBKRTFFWDDCQLH
|
8.5 | IC50 | 2 | — | |
SSJBSCHXKMORSU
|
8.5 | IC50 | 4 | — | |
UGODXHKPBLIJKJ
|
8.5 | IC50 | 4 | — | |
UTPPAOMSIMPNEQ
|
8.5 | IC50 | 4 | — | |
GDJNAASAKVZJNI
|
8.5 | IC50 | 3 | — | |
GEMNVMUNTRERDJ
|
8.5 | IC50 | 2 | — | |
AOILZWVIBHVMLR
|
8.5 | IC50 | 4 | — | |
BNAARZMMBWGEGG
|
8.5 | IC50 | 4 | — | |
GDFZQTWVTPRZJP
|
8.5 | IC50 | 4 | — | |
HQMSWMADUGUYFF
|
8.5 | IC50 | 4 | — | |
HZJTYICHFKEZPB
|
8.5 | IC50 | 4 | — | |
JPMVRYCJGBFRDG
|
8.5 | IC50 | 4 | — | |
MAIZEWVIGRBICN
|
8.5 | IC50 | 4 | — | |
ONJXTGCXZBTXRY
|
8.5 | IC50 | 4 | — | |
QHBNTQCVLLJAGG
|
8.5 | IC50 | 4 | — | |
IDQYDZHQPMPCHM
|
8.5 | IC50 | 4 | — | |
LBWBNPCQUXPCDH
|
8.5 | IC50 | 4 | — | |
ZPWHTTHPHDTDRY
|
8.5 | IC50 | 3 | — | |
BONBXBPLENOTTM
|
8.5 | IC50 | 4 | — | |
BONBXBPLENOTTM
|
8.5 | IC50 | 3 | — | |
NAAAZTBWVPSSHE
|
8.5 | IC50 | 4 | — | |
PTRVZEMPNWFZEI
|
8.5 | IC50 | 4 | — | |
KJLMCBXHAQXCDZ
|
8.5 | IC50 | 4 | — | |
PGXKVCTXUZHTHO
|
8.5 | IC50 | 4 | — | |
QDCNDOVOAIZYTL
|
8.5 | IC50 | 4 | — | |
QDCNDOVOAIZYTL
|
8.5 | IC50 | 4 | — | |
TWBJKVMWEQKJFY
|
8.5 | IC50 | 2 | — | |
YAXKZYIBIZYKIR
|
8.5 | IC50 | 4 | — | |
GBDADLBKHYUAQL
|
8.4 | IC50 | 2 | — | |
IVQYTNHIHIIOCN
|
8.4 | IC50 | 5 | — | |
KTEIFNKAUNYNJU
|
8.4 | Kd | 114 | — | |
WDLJSYMVGMNFSD
|
8.4 | IC50 | 4 | — | |
XJVOXPBGMZCIJM
|
8.4 | IC50 | 2 | — | |
XZEKGVVKPPJAPK
|
8.4 | IC50 | 2 | — | |
MKUAZUIGYWTRKA
|
8.4 | IC50 | 4 | — | |
SUEWBPGMSMAJTQ
|
8.4 | IC50 | 4 | — | |
FRUDSLHJWXUHFH
|
8.4 | IC50 | 3 | — | |
HLKNAIHDOGWCMT
|
8.4 | IC50 | 2 | — | |
RAPSXYUJSKOFLB
|
8.4 | IC50 | 4 | — | |
UVBALELUPGCHKQ
|
8.4 | IC50 | 4 | — | |
XYSYRHAUHUPOHK
|
8.4 | IC50 | 3 | — | |
DXHZDRZKMSATCC
|
8.4 | IC50 | 4 | — | |
KOWRWJFANSWOCN
|
8.4 | IC50 | 4 | — | |
MDBQDUFVZUXGHO
|
8.4 | IC50 | 4 | — | |
MFMGCNRBRYJVAT
|
8.4 | IC50 | 4 | — | |
TTZSNFLLYPYKIL
|
8.4 | IC50 | 7 | — | |
UBUCCNWQOAYWFT
|
8.4 | IC50 | 4 | — | |
VPDVHIDCAMWQER
|
8.4 | IC50 | 4 | — | |
DKLRVMHGCQHXBG
|
8.4 | IC50 | 3 | — | |
HSYSSKFCQHXOBP
|
8.4 | IC50 | 3 | — |