Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QJYWNLGATZHNCX
|
8.6 | IC50 | 4 | — | |
RXKJTHMWVQQQRO
|
8.6 | IC50 | 4 | — | |
SXOGNSSKJOUDNZ
|
8.6 | IC50 | 4 | — | |
WUHGCCVXBHUUSZ
|
8.6 | IC50 | 4 | — | |
XGWKKUQOFQDOKM
|
8.6 | IC50 | 3 | — | |
ZAPJKVKBAKZIMU
|
8.6 | IC50 | 4 | — | |
AOILZWVIBHVMLR
|
8.6 | IC50 | 4 | — | |
KDYGVGVZGXBONW
|
8.6 | IC50 | 4 | — | |
NSYLBOUGDLOZHC
|
8.6 | IC50 | 2 | — | |
QLBFPPCIKGUBAH
|
8.6 | IC50 | 4 | — | |
UMHCVDDSESEXLS
|
8.6 | IC50 | 4 | — | |
VXENEMCDVCFWGW
|
8.6 | IC50 | 3 | — | |
FCDFAUPFHSOSFR
|
8.6 | IC50 | 4 | — | |
MASPYCIEHQXHEE
|
8.6 | IC50 | 4 | — | |
MUSCNFZYEUAAPG
|
8.6 | IC50 | 3 | — | |
ROIWAJLBBPZORU
|
8.6 | IC50 | 4 | — | |
VZOFLHLWMKWZHW
|
8.6 | IC50 | 4 | — | |
ZXSGJKRDMSVFSU
|
8.6 | IC50 | 3 | — | |
ATNAJZHNVLANKY
|
8.6 | IC50 | 4 | — | |
FSEJTXYPUWBYGR
|
8.6 | IC50 | 4 | — | |
IKQPJOFHAZFMNC
|
8.6 | IC50 | 4 | — | |
IUTWSTURTCLHKX
|
8.6 | IC50 | 4 | — | |
KMDUVZLDXOHFPQ
|
8.6 | IC50 | 4 | — | |
SAVZKBLDLPHYOO
|
8.6 | IC50 | 4 | — | |
MJSHVHLADKXCML
|
8.6 | IC50 | 11 | — | |
GHZOFMBOCOPIGL
|
8.6 | IC50 | 2 | — | |
ITRYMWSQXXWWJF
|
8.6 | IC50 | 4 | — | |
OHFCYJVNUVCECF
|
8.6 | IC50 | 4 | — | |
YUKVQCUADDDWFR
|
8.6 | IC50 | 2 | — | |
YVAPXKWBCBCTDS
|
8.6 | IC50 | 3 | — | |
YVAPXKWBCBCTDS
|
8.6 | IC50 | 4 | — | |
ZHQZACQNPQRBGO
|
8.6 | IC50 | 4 | — | |
ATIWZLMXSXMEDE
|
8.5 | IC50 | 2 | — | |
OGEBRHQLRGFBNV
|
8.5 | IC50 | 3 | — | |
OGEBRHQLRGFBNV
|
8.5 | IC50 | 3 | — | |
ORIMXTQTVHCGIW
|
8.5 | IC50 | 4 | — | |
PBLCTGOWTVQZHF
|
8.5 | IC50 | 2 | — | |
RRGONMPXYOQEDE
|
8.5 | IC50 | 4 | — | |
YCNFDYPECZUZNM
|
8.5 | IC50 | 4 | — | |
ZMXXPABXSZBSGM
|
8.5 | IC50 | 4 | — | |
ZOHLAZXVTPODGE
|
8.5 | IC50 | 4 | — | |
LZOJVTCTBSNNNT
|
8.5 | IC50 | 4 | — | |
RIXYJFUGGXKHPG
|
8.5 | IC50 | 4 | — | |
SSJIQTZEUSHBBQ
|
8.5 | IC50 | 4 | — | |
WLJALOYLOJDZQW
|
8.5 | IC50 | 4 | — | |
WMWHVTDZNIVNIE
|
8.5 | IC50 | 9 | — | |
WMWHVTDZNIVNIE
|
8.5 | IC50 | 9 | — | |
CBJZWQSCZBRXDC
|
8.5 | IC50 | 4 | — | |
FXTJCTYAPOCFAC
|
8.5 | IC50 | 4 | — | |
RKITWCYZEAAJLC
|
8.5 | IC50 | 4 | — |