Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KVOOIXIMILKHSX
|
6.2 | IC50 | 2 | — | |
LVMCQNRIJXVCOS
|
6.2 | IC50 | 2 | — | |
NMCDJZKJPUDTBD
|
6.2 | IC50 | 2 | — | |
SDUVWEQOIYQSRO
|
6.2 | IC50 | 2 | — | |
SUGDHXMPLXNQCH
|
6.2 | IC50 | 2 | — | |
WPOIBEJAMKTRNC
|
6.2 | IC50 | 2 | — | |
ZRDFYRNZGRYVBF
|
6.2 | IC50 | 2 | — | |
RFBIIBVIVNVJSA
|
6.2 | IC50 | 2 | — | |
HHFBDROWDBDFBR
|
6.1 | Kd | 40 | Yes | |
IQOCOGQTLHXQMU
|
6.1 | IC50 | 2 | — | |
JZRMSULPXPLESF
|
6.1 | IC50 | 2 | — | |
HMLAOGYJGKIMSB
|
6.1 | IC50 | 2 | — | |
HMPVOPPEDSHUFT
|
6.1 | IC50 | 2 | — | |
HTGGWBJDPLPEPS
|
6.1 | IC50 | 2 | — | |
NAOHATQHGKGARO
|
6.1 | IC50 | 2 | — | |
NJPNCUKTBVUHBB
|
6.1 | IC50 | 2 | — | |
RWHHZRIUWKYUJA
|
6.1 | IC50 | 2 | — | |
YFHWTHUFKDLCHI
|
6.1 | IC50 | 2 | — | |
YYLKKYCXAOBSRM
|
6.1 | Kd | 191 | — | |
ZYYBPQOUQVKJNI
|
6.1 | IC50 | 2 | — | |
GFETUQKKOOEAQJ
|
6.1 | IC50 | 2 | — | |
JOOXLOJCABQBSG
|
6.1 | Kd | 139 | — | |
JREIMVGWCLAHOC
|
6.1 | IC50 | 2 | — | |
PKCOJEQPEFFMMK
|
6.1 | IC50 | 2 | — | |
FTUDPMMKHAMLKT
|
6.1 | IC50 | 3 | — | |
QKJUNBIPFNGGAT
|
6.1 | IC50 | 3 | — | |
TVGHZVBEWSTROH
|
6.1 | IC50 | 2 | — | |
WYCSYGHXJGVXDE
|
6.1 | IC50 | 2 | — | |
KZWSQDIHXXAHML
|
6.1 | IC50 | 2 | — | |
MPVGZUGXCQEXTM
|
6.1 | Kd | 61 | Yes | |
RUKNGDZXNOSJCJ
|
6.1 | IC50 | 2 | — | |
ILTRGYHQTNEKOS
|
6.0 | IC50 | 2 | — | |
MVHPGOCNSYOLJS
|
6.0 | IC50 | 2 | — | |
RSIRXFZBWSKWOR
|
6.0 | IC50 | 3 | — | |
WSJDAGGMIFURQV
|
6.0 | IC50 | 2 | — | |
RFMIJZBBECZAQC
|
6.0 | IC50 | 2 | — | |
AAKJLRGGTJKAMG
|
6.0 | Kd | 50 | Yes | |
PXWBFLDNKAECRK
|
6.0 | IC50 | 2 | — | |
YYDHXOVJKJQURC
|
6.0 | IC50 | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |