Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SDZOULNKJGWLJC
|
6.3 | IC50 | 2 | — | |
SKCNQXHSXCOEQN
|
6.3 | IC50 | 2 | — | |
SRWSOVXHPNAAOR
|
6.3 | IC50 | 2 | — | |
SUXREGNCXSXOFZ
|
6.3 | IC50 | 2 | — | |
TXZRIDXMQZUDMK
|
6.3 | IC50 | 3 | — | |
UBRTVWBFPUFTFQ
|
6.3 | IC50 | 2 | — | |
UISXPDDNFOZHMW
|
6.3 | IC50 | 2 | — | |
USTZAESKZVOYQN
|
6.3 | IC50 | 2 | — | |
VBCRGRNOINTVFO
|
6.3 | IC50 | 2 | — | |
VEOCIRAZZKBKKO
|
6.3 | IC50 | 2 | — | |
VOQFOXNRZJPJLE
|
6.3 | IC50 | 2 | — | |
VQNCJQLQTVPNFF
|
6.3 | IC50 | 2 | — | |
WHRFEMZKPOYXJP
|
6.3 | IC50 | 2 | — | |
WHXBKUCRLXDOGL
|
6.3 | IC50 | 2 | — | |
WNKZIEUWVPWSJA
|
6.3 | IC50 | 2 | — | |
WYSKAJAOYHAYCD
|
6.3 | IC50 | 2 | — | |
WYSKAJAOYHAYCD
|
6.3 | IC50 | 2 | — | |
XEGPHZMYVJLNIO
|
6.3 | IC50 | 3 | — | |
YBCVPFLUANOFHV
|
6.3 | IC50 | 3 | — | |
YBROIBYJRIQHTK
|
6.3 | IC50 | 2 | — | |
YFWVUIYRHIEOSI
|
6.3 | IC50 | 2 | — | |
YKNIFWRCNVOETK
|
6.3 | IC50 | 2 | — | |
ZETHWMVNIMDCLY
|
6.3 | IC50 | 2 | — | |
ZGOBWUJNSGWNHI
|
6.3 | IC50 | 2 | — | |
ZJQBGCUUGXCPKJ
|
6.3 | IC50 | 2 | — | |
ZSPYZKJALVPWOV
|
6.3 | IC50 | 2 | — | |
CSWIFIVPMHAOGX
|
6.2 | IC50 | 2 | — | |
QBRQTJMZEYORSP
|
6.2 | Kd | 12 | — | |
ODHHBTQTAVNJQP
|
6.2 | IC50 | 2 | — | |
RQMXEHSOMYFNKM
|
6.2 | IC50 | 2 | — | |
YSEOULVZPWEYPN
|
6.2 | IC50 | 2 | — | |
NPPNDOYKLAXXAS
|
6.2 | IC50 | 2 | — | |
KKAICBOHJLVDCE
|
6.2 | IC50 | 2 | — | |
QJBBRIGNNQUHMN
|
6.2 | IC50 | 2 | — | |
NDBJFFCSTXBTFV
|
6.2 | IC50 | 6 | — | |
MMJWZGGVKOHMPQ
|
6.2 | IC50 | 6 | — | |
NBKAWHPTEZYULQ
|
6.2 | IC50 | 2 | — | |
PMCFVEARPWIGJR
|
6.2 | IC50 | 2 | — | |
QLRMYWGPTHTIEO
|
6.2 | IC50 | 2 | — | |
XSXUZWJPMJGSJV
|
6.2 | IC50 | 2 | — | |
XYASHXPUZJDWIO
|
6.2 | IC50 | 7 | — | |
JQQNLXLUEMOKQW
|
6.2 | IC50 | 2 | — | |
BWPIHLJJXPJVRB
|
6.2 | IC50 | 2 | — | |
CXIPPVQDQRFLFI
|
6.2 | IC50 | 2 | — | |
FKWHTFASCNDJAH
|
6.2 | IC50 | 2 | — | |
FLXFUGYYZDJYLE
|
6.2 | IC50 | 2 | — | |
GYLJUKWLPMHVRN
|
6.2 | IC50 | 2 | — | |
HPXOEJIGVHSELH
|
6.2 | IC50 | 2 | — | |
HUORQQWKJRLEPT
|
6.2 | IC50 | 2 | — | |
JPZHJBRLZGPDAW
|
6.2 | IC50 | 2 | — |