Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DRLDUGDBHRWAGE
|
6.3 | IC50 | 2 | — | |
DRWFPMANDOOIDL
|
6.3 | IC50 | 2 | — | |
DTKKTUUDABIULF
|
6.3 | IC50 | 3 | — | |
DZGNYCKQISDLDR
|
6.3 | IC50 | 2 | — | |
DZGNYCKQISDLDR
|
6.3 | IC50 | 2 | — | |
FDZKCGQKBRGCHT
|
6.3 | IC50 | 2 | — | |
FKEIYILKGUQVFR
|
6.3 | IC50 | 2 | — | |
FWILABWFWCXXHH
|
6.3 | IC50 | 2 | — | |
FXECSFGCDPHDIV
|
6.3 | IC50 | 2 | — | |
GFNQZVJUGWXFOR
|
6.3 | IC50 | 2 | — | |
GHJOPDWWDYLDPQ
|
6.3 | IC50 | 2 | — | |
GHYJHXVIHGZWLO
|
6.3 | IC50 | 2 | — | |
GKKRAVYWSLIBMJ
|
6.3 | IC50 | 2 | — | |
GRJHFCOVFFKFSJ
|
6.3 | IC50 | 2 | — | |
HBENISDMECHQSQ
|
6.3 | IC50 | 3 | — | |
IAFDYYBXGULYAS
|
6.3 | IC50 | 2 | — | |
IIQJYPYTLGEBIE
|
6.3 | IC50 | 2 | — | |
IZMXTWYXRXNDPN
|
6.3 | IC50 | 2 | — | |
JHCORCZCAFONIQ
|
6.3 | IC50 | 2 | — | |
JJAHVHNFADQPQV
|
6.3 | IC50 | 2 | — | |
JOEJPJLBUUYFKP
|
6.3 | IC50 | 2 | — | |
JSYUPEDNWUOTAB
|
6.3 | IC50 | 2 | — | |
JZWMOYVAUTWRAA
|
6.3 | IC50 | 2 | — | |
KFZQJQMKXCKADU
|
6.3 | IC50 | 2 | — | |
KOGINFSZWQZUSG
|
6.3 | IC50 | 3 | — | |
KVLVPMNDRHOZLP
|
6.3 | IC50 | 2 | — | |
KZYNSZVLJLXZEZ
|
6.3 | IC50 | 2 | — | |
LOODYZPMRGPWCF
|
6.3 | IC50 | 2 | — | |
LUVKMLLQMCZBGO
|
6.3 | IC50 | 2 | — | |
MQHBJQJKPRSJRX
|
6.3 | IC50 | 2 | — | |
MWSLVORBGRTVRI
|
6.3 | IC50 | 2 | — | |
MYPUPNZFDCNJSA
|
6.3 | IC50 | 2 | — | |
MYUJBDVTLXXMHN
|
6.3 | IC50 | 3 | — | |
NEHBMIAYXIRHIO
|
6.3 | IC50 | 2 | — | |
NNAPEAGXVRJCIQ
|
6.3 | IC50 | 2 | — | |
NOWQREWVISHNOQ
|
6.3 | IC50 | 2 | — | |
NRWZOZHFNIXRFZ
|
6.3 | IC50 | 2 | — | |
OHAAFYYZLAILTE
|
6.3 | IC50 | 2 | — | |
ORMXEYBLYMZYLP
|
6.3 | IC50 | 2 | — | |
OTKTYQXOBFJYGG
|
6.3 | IC50 | 3 | — | |
OXTIJGNQHLIQQQ
|
6.3 | IC50 | 2 | — | |
PAJRSBHPHKZQCV
|
6.3 | IC50 | 2 | — | |
PTCNXTACPMUJGC
|
6.3 | IC50 | 3 | — | |
QABDFIDZXJGZPC
|
6.3 | IC50 | 2 | — | |
QKLHJJJNGDFUIT
|
6.3 | IC50 | 3 | — | |
QRIVXCKMXGMYSA
|
6.3 | IC50 | 3 | — | |
QWMQKEAUBCSAHZ
|
6.3 | IC50 | 2 | — | |
RAPKAHFDNKOYTF
|
6.3 | IC50 | 3 | — | |
RPHAHGRSQTZHAE
|
6.3 | IC50 | 2 | — | |
RQOFQPPGGQJMHO
|
6.3 | IC50 | 2 | — |