Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FLEDZRUQPMPOFA
|
8.8 | IC50 | 4 | — | |
IMQXMHYXTAYQDO
|
8.8 | IC50 | 3 | — | |
JGIUBJWBTUOQHP
|
8.8 | IC50 | 4 | — | |
LFOWPAZJQIZNHI
|
8.8 | IC50 | 4 | — | |
LFOWPAZJQIZNHI
|
8.8 | IC50 | 4 | — | |
LOJVVUQLHLHRMD
|
8.8 | IC50 | 3 | — | |
PINVBZQZBYOHQT
|
8.8 | IC50 | 2 | — | |
RGAZVGZUBCFHRJ
|
8.8 | IC50 | 5 | — | |
RPXUPQNHYGEYEU
|
8.8 | IC50 | 4 | — | |
ZVGXWQWGKFNZAK
|
8.8 | IC50 | 4 | — | |
MIOQFVQXGRHCSR
|
8.8 | IC50 | 4 | — | |
MUIPWSHBCRIWKJ
|
8.8 | IC50 | 4 | — | |
NVHUKBRGAIBVPK
|
8.8 | IC50 | 4 | — | |
QBBXSRZGLKRAMO
|
8.8 | IC50 | 4 | — | |
UIKRXGNEQUHBIX
|
8.8 | IC50 | 4 | — | |
WQLWLOMHWYQNFN
|
8.8 | IC50 | 3 | — | |
WQLWLOMHWYQNFN
|
8.8 | IC50 | 4 | — | |
HSYSSKFCQHXOBP
|
8.7 | IC50 | 4 | — | |
IEXXROGGKUBLPS
|
8.7 | IC50 | 4 | — | |
JNYMZWUOQWXOII
|
8.7 | IC50 | 3 | — | |
KIMZAWNVESXXES
|
8.7 | IC50 | 2 | — | |
TUSFBIZKPNHLKT
|
8.7 | IC50 | 4 | — | |
AJLUXNJECIAQBR
|
8.7 | IC50 | 4 | — | |
CREINZJAYXIGBI
|
8.7 | IC50 | 4 | — | |
HFOSJCQJOTUBNX
|
8.7 | IC50 | 2 | — | |
KFXRRWQDJNJMKE
|
8.7 | IC50 | 4 | — | |
PHXDBKCVMGZILA
|
8.7 | IC50 | 2 | — | |
PZOHZBXMRBOYRF
|
8.7 | IC50 | 2 | — | |
XQTQDOHPJHEUPU
|
8.7 | IC50 | 2 | — | |
PWNYLFPOEAFAPH
|
8.7 | IC50 | 2 | — | |
FPLGAASDZAAKLR
|
8.7 | IC50 | 2 | — | |
MAHJDNICCJZVKW
|
8.7 | IC50 | 4 | — | |
SERBYZUNBVTZJZ
|
8.7 | IC50 | 3 | — | |
WBAXZSZODFIDGK
|
8.7 | IC50 | 4 | — | |
YTEDDIJNHJDCLR
|
8.7 | IC50 | 4 | — | |
HBQLAXMLLMAJCM
|
8.7 | IC50 | 4 | — | |
IJBQYPBBOUFSEN
|
8.7 | IC50 | 3 | — | |
SLRXPNTXSLSWEL
|
8.7 | IC50 | 2 | — | |
YWILRIPPYUJHMX
|
8.7 | IC50 | 4 | — | |
BPOGHKOSOWZBGZ
|
8.7 | IC50 | 4 | — | |
DBAIZGMGQSAOER
|
8.7 | IC50 | 2 | — | |
PXHDQHNAGHIZGO
|
8.7 | IC50 | 4 | — | |
QEAUPAREISBURF
|
8.7 | IC50 | 4 | — | |
VHIPJRRFLDFKSD
|
8.7 | IC50 | 4 | — | |
YKSFAELRDYTAHZ
|
8.7 | IC50 | 3 | — | |
DYQYODJNEBRPRK
|
8.6 | IC50 | 4 | — | |
FWXIWEQAGQKYSB
|
8.6 | IC50 | 4 | — | |
IAURWWSIIMOBHU
|
8.6 | IC50 | 4 | — | |
LLDMPYKKTBBIRQ
|
8.6 | IC50 | 3 | — | |
LOMPHWBCBDXNOY
|
8.6 | IC50 | 4 | — |