Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UBRFJUHJYBVBTP
|
6.5 | IC50 | 2 | — | |
VAAUYOSCIMZUKR
|
6.5 | IC50 | 3 | — | |
VZDLPJYBPUCWAE
|
6.5 | IC50 | 2 | — | |
WPQIUKYVSOXPET
|
6.5 | IC50 | 2 | — | |
WSBMMJILOSMNBS
|
6.5 | IC50 | 2 | — | |
XWJPJDSYKZCYMC
|
6.5 | IC50 | 2 | — | |
YKCROARFPLKWJI
|
6.5 | IC50 | 2 | — | |
ZJEXDIVRZSPIDL
|
6.5 | IC50 | 3 | — | |
BHQBNRDVYQVMDL
|
6.4 | IC50 | 2 | — | |
ODPGGGTTYSGTGO
|
6.4 | Kd | 153 | — | |
OQRDMLSFWXYGCO
|
6.4 | IC50 | 2 | — | |
FCOQUZVLXLTSQN
|
6.4 | IC50 | 2 | — | |
JWNPDZNEKVCWMY
|
6.4 | Kd | 57 | Yes | |
IEJMTNVTRDPUHP
|
6.4 | IC50 | 2 | — | |
OQLLSZTVSXCTIX
|
6.4 | IC50 | 2 | — | |
ZRRDEVCMPKUGEA
|
6.4 | IC50 | 2 | — | |
UFBWCXYTJNSQAR
|
6.3 | IC50 | 2 | — | |
BKCJISRRNROAEV
|
6.3 | IC50 | 2 | — | |
SHPFDGWALWEPGS
|
6.3 | Kd | 35 | — | |
UFGKRFSRVWAORW
|
6.3 | IC50 | 2 | — | |
ADELQQCPARGKLR
|
6.3 | IC50 | 2 | — | |
NJKNVLHXHQQCKI
|
6.3 | IC50 | 2 | — | |
WIVPSHFRGVZOQV
|
6.3 | IC50 | 2 | — | |
SIXVRXARNAVBTC
|
6.3 | IC50 | 12 | — | |
UGPDJIJFANODJH
|
6.3 | IC50 | 12 | — | |
LJCANGDUIWZUBX
|
6.3 | IC50 | 2 | — | |
WSXGWGXVUJHSDF
|
6.3 | IC50 | 2 | — | |
WYEUDIXCTGHYOQ
|
6.3 | IC50 | 2 | — | |
CGTZBMSJBJIXFU
|
6.3 | IC50 | 2 | — | |
CQHNWEKZZSCARI
|
6.3 | IC50 | 2 | — | |
JXMVPCLSCZWMLY
|
6.3 | IC50 | 2 | — | |
VVQFSZLHAOOPPI
|
6.3 | IC50 | 2 | — | |
YWPWDZZAROUKLO
|
6.3 | IC50 | 2 | — | |
DYXYAJUTMZMYSZ
|
6.3 | IC50 | 2 | — | |
RJSUQBZTJGZMTH
|
6.3 | IC50 | 2 | — | |
UKPKGXOPGQHRRJ
|
6.3 | IC50 | 2 | — | |
AGSNFEMFMGJZFO
|
6.3 | IC50 | 2 | — | |
AMQOJYCRTWTXKW
|
6.3 | IC50 | 2 | — | |
BAGLRIYGLUAGSG
|
6.3 | IC50 | 3 | — | |
BJCSBDZHBPODPN
|
6.3 | IC50 | 2 | — | |
BUXYDKZKYRETLE
|
6.3 | IC50 | 2 | — | |
BVQOQCVSTRWIJJ
|
6.3 | IC50 | 2 | — | |
BYOPTHRZGQDQRO
|
6.3 | IC50 | 2 | — | |
CCYBRUQGEAOPNW
|
6.3 | IC50 | 2 | — | |
CFNVHHHXPVFHNU
|
6.3 | IC50 | 2 | — | |
CGGBWSCTIMLZPY
|
6.3 | IC50 | 2 | — | |
CIZMHSSVMQOOSL
|
6.3 | IC50 | 2 | — | |
COZPNRXVDFBHEC
|
6.3 | IC50 | 2 | — | |
DMHSZFIBOGIPRH
|
6.3 | IC50 | 2 | — | |
DPYYQWWXBGMVOA
|
6.3 | IC50 | 2 | — |