Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SZVQFUFNMUBFOE
|
6.6 | IC50 | 2 | — | |
UGLZXRPFZYUMAE
|
6.6 | IC50 | 2 | — | |
XPJNWRLQVHKGRY
|
6.6 | IC50 | 2 | — | |
YNXHDCOYJGXDDO
|
6.6 | IC50 | 2 | — | |
YZXPXXZCCJVPRH
|
6.6 | IC50 | 3 | — | |
JCRDCMIKTSPWHJ
|
6.5 | IC50 | 2 | — | |
JXIOZYRODOOPLU
|
6.5 | IC50 | 2 | — | |
PHACAAIWJAWPHA
|
6.5 | IC50 | 2 | — | |
HBEYTTVTDWYNAA
|
6.5 | IC50 | 2 | — | |
HDAXKYDWUMHJMD
|
6.5 | IC50 | 2 | — | |
KTBSXLIQKWEBRB
|
6.5 | IC50 | 7 | — | |
LBFOYYYOENDKSM
|
6.5 | IC50 | 3 | — | |
LLZWKZMRVJFITC
|
6.5 | IC50 | 3 | — | |
MYBMVTCYUBVOEK
|
6.5 | IC50 | 2 | — | |
PHXVZSVYYRTVHM
|
6.5 | IC50 | 2 | — | |
PUNWZJKAQIQKQL
|
6.5 | IC50 | 2 | — | |
QFPGZAJRDFHPCE
|
6.5 | IC50 | 3 | — | |
VCJFOLMEZCAWFO
|
6.5 | IC50 | 3 | — | |
VQDFOOLMNPPTBD
|
6.5 | IC50 | 3 | — | |
WQXUGBZSZWSUTM
|
6.5 | IC50 | 3 | — | |
XWGQRTQXVAWLEI
|
6.5 | IC50 | 3 | — | |
GLOKAXXDXBXLRH
|
6.5 | IC50 | 2 | — | |
XMLHEOBAISADLD
|
6.5 | IC50 | 2 | — | |
XMZOHULIEPXEFI
|
6.5 | IC50 | 2 | — | |
YQDQJTHWHPDCGQ
|
6.5 | IC50 | 2 | — | |
FECSXNXXQKGAJO
|
6.5 | IC50 | 3 | — | |
GIVXEVXCESBALN
|
6.5 | IC50 | 2 | — | |
JXOOCVOCZKLKCJ
|
6.5 | IC50 | 2 | — | |
CZNWNZFIYBTRPU
|
6.5 | IC50 | 2 | — | |
ATBDIPDCACEXQS
|
6.5 | IC50 | 2 | — | |
BTLGQUCTPQAVFE
|
6.5 | IC50 | 3 | — | |
CKMFFVUKUWSUSB
|
6.5 | IC50 | 2 | — | |
CQEFDVMDIZEGMM
|
6.5 | IC50 | 3 | — | |
GBHAWNHMHWSXOP
|
6.5 | IC50 | 3 | — | |
IVKPXXIBAHRJLH
|
6.5 | IC50 | 3 | — | |
IWQUQHHOHMTSSG
|
6.5 | IC50 | 2 | — | |
JIRPGDPVSYXTQB
|
6.5 | IC50 | 3 | — | |
KQFRLAVHFVOCHP
|
6.5 | IC50 | 3 | — | |
LKKVMNQKZUOIIS
|
6.5 | IC50 | 2 | — | |
LLXTYNLCGJXTSA
|
6.5 | IC50 | 3 | — | |
LZXUNBCSKDGSRW
|
6.5 | IC50 | 2 | — | |
MNMBZMNBJGWCOY
|
6.5 | IC50 | 3 | — | |
MTEGSTLSVBUGPL
|
6.5 | IC50 | 3 | — | |
ODXMRLSGGABXAR
|
6.5 | IC50 | 2 | — | |
OOGRPSIRCBIFAB
|
6.5 | IC50 | 3 | — | |
OZDGFJODPAGVGR
|
6.5 | IC50 | 2 | — | |
QFDWIEDSPKSMIC
|
6.5 | IC50 | 2 | — | |
RQNZLJJIYKQXOF
|
6.5 | IC50 | 2 | — | |
SXMIOBCJEWYZCT
|
6.5 | IC50 | 2 | — | |
TVLLCZBDUVKPOT
|
6.5 | IC50 | 2 | — |