Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AWJXWMJXQDNNHI
|
6.6 | IC50 | 3 | — | |
AYAAYSFAENPXLJ
|
6.6 | IC50 | 3 | — | |
BAXYAPSMRBNZRD
|
6.6 | IC50 | 2 | — | |
BJHLJRKGOCSNAB
|
6.6 | IC50 | 2 | — | |
DZKHRKMBAPEIOK
|
6.6 | IC50 | 2 | — | |
FNYWKJPMFGZVAH
|
6.6 | IC50 | 2 | — | |
FSVJWBPBIXGNJR
|
6.6 | IC50 | 2 | — | |
GCEHBYASKOQVGC
|
6.6 | IC50 | 2 | — | |
GFUCPRWCLHVWDC
|
6.6 | IC50 | 2 | — | |
GJLXMTNNDQGGKD
|
6.6 | IC50 | 2 | — | |
GQLITRCSLFCUTG
|
6.6 | IC50 | 2 | — | |
IJXRHXHFJDIXQV
|
6.6 | IC50 | 2 | — | |
IMTPDXPBIHKJMT
|
6.6 | IC50 | 2 | — | |
IRDLISIFNYBKFQ
|
6.6 | IC50 | 2 | — | |
JESGNXZGLBLJDC
|
6.6 | IC50 | 2 | — | |
JISOVQKSGVQADF
|
6.6 | IC50 | 2 | — | |
KLKYJRXPXAKVSC
|
6.6 | IC50 | 2 | — | |
LQBDZMZNBNPGIB
|
6.6 | IC50 | 2 | — | |
MTECOFLCYIXTPZ
|
6.6 | IC50 | 2 | — | |
MVHGAHBKSNCJEL
|
6.6 | IC50 | 2 | — | |
NWOWRWKOTHXMFN
|
6.6 | IC50 | 2 | — | |
OEZKMUKPUFZGCU
|
6.6 | IC50 | 2 | — | |
QPXKLICOIXEZHL
|
6.6 | IC50 | 2 | — | |
QUGMULQJKFZKBO
|
6.6 | IC50 | 3 | — | |
RAFWWCIIHOSBCO
|
6.6 | IC50 | 2 | — | |
RIWPMLGHVQKIKL
|
6.6 | IC50 | 2 | — | |
SIISCDRBPBFCTB
|
6.6 | IC50 | 2 | — | |
UKMXSBKKSKVHAG
|
6.6 | IC50 | 2 | — | |
URYRJGMTBZCOOI
|
6.6 | IC50 | 3 | — | |
UTJMZPDAIKTLII
|
6.6 | IC50 | 3 | — | |
WGSRIKGDSWUTBU
|
6.6 | IC50 | 3 | — | |
WOQQMUNLESVVOT
|
6.6 | IC50 | 2 | — | |
YEWUZPDYMNCRNM
|
6.6 | IC50 | 2 | — | |
YNFPEISXYNRRFY
|
6.6 | IC50 | 2 | — | |
YUGVQSDODGIURB
|
6.6 | IC50 | 2 | — | |
YZBOIOWUBUUXNT
|
6.6 | IC50 | 3 | — | |
ZPTOECURBRGDME
|
6.6 | IC50 | 3 | — | |
ZXWHXKOLSGGTQX
|
6.6 | IC50 | 3 | — | |
SYXAZEFBEOQPCZ
|
6.6 | Kd | 3 | — | |
BQOPPXMDAUTYSM
|
6.6 | IC50 | 2 | — | |
VEDWRPNOJNKGOL
|
6.6 | IC50 | 2 | — | |
YLKNZRZBRWCKRM
|
6.6 | IC50 | 2 | — | |
YLKPPBUPVVBPDB
|
6.6 | IC50 | 2 | — | |
BGSWWJPEXPOCRJ
|
6.6 | IC50 | 2 | — | |
COFZOFHLQQEYAH
|
6.6 | IC50 | 2 | — | |
FQDAGUFKVOIFKE
|
6.6 | IC50 | 2 | — | |
FWKPMQSKTCDKAE
|
6.6 | IC50 | 3 | — | |
GVWDYJCKQRURCQ
|
6.6 | IC50 | 3 | — | |
IPPTWJWXDUGTIB
|
6.6 | IC50 | 3 | — | |
QZXMHSSMITURNJ
|
6.6 | IC50 | 2 | — |