Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RWHXYPTULXPVSO
|
6.8 | IC50 | 2 | — | |
YTXPYXBASKYQMU
|
6.8 | IC50 | 2 | — | |
BBEKTQZNBOIUQG
|
6.8 | IC50 | 2 | — | |
ZHJHMBLIFHFWBT
|
6.8 | IC50 | 2 | — | |
NLEBCCQURQQOSU
|
6.7 | IC50 | 2 | — | |
RENRJGXFTHYPPG
|
6.7 | IC50 | 2 | — | |
RQZDAXOPNDQREW
|
6.7 | IC50 | 2 | — | |
VKLVODAMMAVNIA
|
6.7 | IC50 | 2 | — | |
NBWPBWVCXDBJIJ
|
6.7 | IC50 | 2 | — | |
XJQJAMKWRLSFRE
|
6.7 | IC50 | 2 | — | |
AGPYHKUKKNTOOF
|
6.7 | IC50 | 2 | — | |
MGETVYBTJTWGJG
|
6.7 | IC50 | 2 | — | |
SAIJSXPUPZBTMI
|
6.7 | IC50 | 2 | — | |
WRJXNDZLDVGDIF
|
6.7 | IC50 | 2 | — | |
XQLXHIGCGPBKTR
|
6.7 | Kd | 5 | — | |
YJZTUFCHNMWPJK
|
6.7 | IC50 | 2 | — | |
HKBYHKNYHRHQLA
|
6.7 | IC50 | 2 | — | |
XCXMZUYZFOFSTB
|
6.7 | IC50 | 2 | — | |
BJFADWIVXIPKGC
|
6.7 | IC50 | 2 | — | |
FGQUZTPOBIQTMT
|
6.7 | IC50 | 2 | — | |
GAYKTWZLTBSKSY
|
6.7 | IC50 | 2 | — | |
GQTGXSGWXVDRDZ
|
6.7 | IC50 | 2 | — | |
JCWYTIFWSKODPB
|
6.7 | IC50 | 2 | — | |
JJKGYGMFHAYASJ
|
6.7 | IC50 | 3 | — | |
KGFCIMCRXWIOFT
|
6.7 | IC50 | 2 | — | |
MIEQOSSLRLYSHP
|
6.7 | IC50 | 2 | — | |
NAXVZCLZSQGACR
|
6.7 | IC50 | 2 | — | |
OAQLTCVWCQRWEW
|
6.7 | IC50 | 2 | — | |
ULIRDGCRHUZAAA
|
6.7 | IC50 | 2 | — | |
BJFADWIVXIPKGC
|
6.7 | IC50 | 2 | — | |
PHYBXPXVBJFNTE
|
6.7 | IC50 | 2 | — | |
YLSAFDQGYSUAFT
|
6.7 | IC50 | 2 | — | |
HQVPDRIYDIRTBE
|
6.7 | IC50 | 2 | — | |
IQIVRGUWXKHLHL
|
6.7 | IC50 | 2 | — | |
ZOEILZXFYPPMTR
|
6.7 | IC50 | 2 | — | |
AUUMOHGHBVZXHF
|
6.7 | IC50 | 2 | — | |
HOXZXBFXGVZLRF
|
6.7 | IC50 | 2 | — | |
VJBZMEXUEJVLAU
|
6.7 | IC50 | 2 | — | |
GHVZTMWFDRXUMG
|
6.6 | IC50 | 2 | — | |
HNAKLVMXRNMVMX
|
6.6 | IC50 | 2 | — | |
RNUHCYHFEQLMQN
|
6.6 | IC50 | 2 | — | |
UBYNKDNUYDOWAR
|
6.6 | IC50 | 2 | — | |
VTXUNTHLMBMYAD
|
6.6 | IC50 | 2 | — | |
YZTURFSBHYCCGX
|
6.6 | IC50 | 2 | — | |
OENGSVYTCJNWNJ
|
6.6 | IC50 | 2 | — | |
LCZJQUXLNMYSLS
|
6.6 | IC50 | 2 | — | |
LGWOKPLTMXFKLZ
|
6.6 | IC50 | 2 | — | |
YINIQNXRRAYBRJ
|
6.6 | IC50 | 2 | — | |
FDBSFRHJILHTNZ
|
6.6 | IC50 | 2 | — | |
AFNUJSJSTUJZNN
|
6.6 | IC50 | 2 | — |