Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BEDLWZIQKBYUTB
|
7.0 | IC50 | 2 | — | |
NUTKAHHQRZGHIS
|
7.0 | IC50 | 2 | — | |
YLSAFDQGYSUAFT
|
7.0 | IC50 | 2 | — | |
MRSQKEXVUFZIMD
|
6.9 | IC50 | 2 | — | |
PCYYUIIBSKPSCD
|
6.9 | IC50 | 2 | — | |
AVDYSPPBTBDYMU
|
6.9 | IC50 | 2 | — | |
JUQPSUXJSPFYGR
|
6.9 | IC50 | 2 | — | |
YPCHDIQOJDQWRM
|
6.9 | IC50 | 2 | — | |
ARRZKLMLWJSTIP
|
6.9 | IC50 | 2 | — | |
AWZRHMXFDZUHLF
|
6.9 | IC50 | 2 | — | |
BQICBFKSXAVIBF
|
6.9 | IC50 | 4 | — | |
NBXADWAEHKGGJP
|
6.9 | IC50 | 2 | — | |
OMLSWMSNQYAKOY
|
6.9 | IC50 | 2 | — | |
XGAALYULZCHKHO
|
6.9 | IC50 | 2 | — | |
AEGRAVKQKLWNSA
|
6.9 | IC50 | 2 | — | |
FSWNWXIANJUKSD
|
6.9 | IC50 | 2 | — | |
KMXWHWXTNYCRNJ
|
6.9 | IC50 | 3 | — | |
LZLIMPWYCRFCKB
|
6.9 | IC50 | 2 | — | |
NGWKXRYBGADMTC
|
6.9 | IC50 | 3 | — | |
PRISLGCTIWIYSJ
|
6.9 | IC50 | 2 | — | |
SKYHCUQSFHNVGB
|
6.9 | IC50 | 2 | — | |
GYWSOFHZIUSHFA
|
6.9 | IC50 | 2 | — | |
IOIMKJTYVDQVKR
|
6.9 | IC50 | 2 | — | |
LVUPJIBJEABNLA
|
6.9 | IC50 | 2 | — | |
AQBVKZHNZSNTDM
|
6.9 | IC50 | 2 | — | |
WTCQJADHNRKLTQ
|
6.9 | IC50 | 2 | — | |
LFNLHBNNYPVNJY
|
6.8 | IC50 | 2 | — | |
ZJTWKNHQHNLTPO
|
6.8 | IC50 | 3 | — | |
UNWQZQOUOXVJKE
|
6.8 | IC50 | 2 | — | |
DYTOVPQOWGLXKV
|
6.8 | IC50 | 3 | — | |
FPQNRXITKTZFMF
|
6.8 | Kd | 13 | — | |
GUZDWCGVMFWILW
|
6.8 | IC50 | 3 | — | |
IYNYCMYPORBQHO
|
6.8 | IC50 | 2 | — | |
OSQTZXWCOXMSCA
|
6.8 | IC50 | 2 | — | |
WOYNBJPVZBBWGG
|
6.8 | IC50 | 2 | — | |
WWFNZSCHGGHKJA
|
6.8 | IC50 | 2 | — | |
HJOCAHLQALFFEI
|
6.8 | IC50 | 3 | — | |
LMKSUPHSUOCPTM
|
6.8 | IC50 | 2 | — | |
LZPFBEBTZBKKFB
|
6.8 | IC50 | 3 | — | |
MCRHIHOQPHSEMM
|
6.8 | IC50 | 2 | — | |
MXFGPNMMPZLQTR
|
6.8 | IC50 | 2 | — | |
OYFAPWKIKGMNQO
|
6.8 | IC50 | 2 | — | |
ASMANSOISNDQDG
|
6.8 | IC50 | 2 | — | |
YBWYETJWZZCBAO
|
6.8 | IC50 | 2 | — | |
ZPWPDCBMIRNATA
|
6.8 | IC50 | 2 | — | |
FSCSEURZUOOESW
|
6.8 | IC50 | 2 | — | |
WGGIKOGLKDIBTL
|
6.8 | IC50 | 2 | — | |
ILONTPDVQVKFCL
|
6.8 | IC50 | 3 | — | |
NHHQJBCNYHBUSI
|
6.8 | Kd | 220 | — | |
RVDBTAAWJRHFHM
|
6.8 | IC50 | 2 | — |