Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TVLLCZBDUVKPOT
|
7.0 | IC50 | 2 | — | |
TYIYGZKYIWNRLG
|
7.0 | IC50 | 3 | — | |
UBPYILGKFZZVDX
|
7.0 | Kd | 130 | Yes | |
UGOMUILQNWWAHA
|
7.0 | IC50 | 3 | — | |
UGXRNWDDMUYEMS
|
7.0 | IC50 | 3 | — | |
UKMYCSRPAHMNQY
|
7.0 | IC50 | 3 | — | |
UQHTVZLEOZKMCJ
|
7.0 | IC50 | 2 | — | |
URVZKSVKISSTJA
|
7.0 | IC50 | 3 | — | |
UXNAQIKBOGDYID
|
7.0 | IC50 | 3 | — | |
VEFBRFNHAWOVSM
|
7.0 | IC50 | 3 | — | |
VENHMKIUHYTQKE
|
7.0 | IC50 | 3 | — | |
VGOUFJFPXAHHOY
|
7.0 | IC50 | 3 | — | |
VICYIZHIHYLSRP
|
7.0 | IC50 | 3 | — | |
VMHNYHNSPZAIKI
|
7.0 | IC50 | 3 | — | |
VNXBUNLANJTOSX
|
7.0 | IC50 | 3 | — | |
VSOINEKSRSZPEM
|
7.0 | IC50 | 3 | — | |
VTHVLRULJMIZBP
|
7.0 | IC50 | 3 | — | |
VVLGFZDIFOANTI
|
7.0 | IC50 | 3 | — | |
WAKOFPSCZPFLKB
|
7.0 | IC50 | 3 | — | |
WAYCKHGOVFVEOO
|
7.0 | IC50 | 2 | — | |
WFFBCQOLUZBHAQ
|
7.0 | IC50 | 3 | — | |
WGNKZRABLXPPLX
|
7.0 | IC50 | 2 | — | |
WMQDFIKSPIVJQC
|
7.0 | IC50 | 3 | — | |
WQURIRYZXSSJJO
|
7.0 | IC50 | 3 | — | |
WSKRUPWLZJJTHT
|
7.0 | IC50 | 2 | — | |
WXXXGQDFKBMVQH
|
7.0 | IC50 | 3 | — | |
XEJLFALBWSEBQR
|
7.0 | IC50 | 3 | — | |
XJWVUJVVTSKKFL
|
7.0 | IC50 | 3 | — | |
XOVPBRHAQXBKEX
|
7.0 | IC50 | 3 | — | |
XRNKKLQKSUGXMM
|
7.0 | IC50 | 2 | — | |
XYVMWPBBCZJSQR
|
7.0 | IC50 | 2 | — | |
YDHWMUFVANAUEA
|
7.0 | IC50 | 2 | — | |
YDPQNYWBOKPIBM
|
7.0 | IC50 | 3 | — | |
YECXZZMXYNBBBT
|
7.0 | IC50 | 3 | — | |
YGIWEFOAKYQLJW
|
7.0 | IC50 | 3 | — | |
YLDJAAQIXCLXGK
|
7.0 | IC50 | 3 | — | |
YLMIZGLXVFMOMS
|
7.0 | IC50 | 3 | — | |
YUEWKPYNHMRLBN
|
7.0 | IC50 | 3 | — | |
ZAFKMBCJTMLVDZ
|
7.0 | IC50 | 3 | — | |
ZATHUJKXAQGLHV
|
7.0 | IC50 | 3 | — | |
ZAVSIGQQWQZRHD
|
7.0 | IC50 | 3 | — | |
ZCKALRAODSTKGS
|
7.0 | IC50 | 2 | — | |
ZHMVEMBLZBGVLQ
|
7.0 | IC50 | 3 | — | |
ZHSWEEUFAGJWSN
|
7.0 | IC50 | 3 | — | |
ZIDWBSKXODQRJU
|
7.0 | IC50 | 3 | — | |
ZPOYSUSBRCQWDE
|
7.0 | IC50 | 3 | — | |
ZRCUBFAHEMHGPQ
|
7.0 | IC50 | 3 | — | |
ZVMGEBXGQJCVMB
|
7.0 | IC50 | 2 | — | |
ZVQCZWRADWOIDU
|
7.0 | IC50 | 3 | — | |
ZWICTTPAXYPCOC
|
7.0 | IC50 | 3 | — |