Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PMVXHUSSOMVCBR
|
7.0 | IC50 | 3 | — | |
PMWOTEZTNPQJII
|
7.0 | IC50 | 3 | — | |
PNYFPUNIXTWPEK
|
7.0 | IC50 | 3 | — | |
POWGNPIDPQTBTI
|
7.0 | IC50 | 3 | — | |
PPUAUWVICIBUPX
|
7.0 | IC50 | 3 | — | |
PQRGSAKVQKBLOB
|
7.0 | IC50 | 3 | — | |
PQRONPGNROKBKK
|
7.0 | IC50 | 3 | — | |
PUBMNVMMPVYBBT
|
7.0 | IC50 | 3 | — | |
PXJNEVPUNYVTHU
|
7.0 | IC50 | 3 | — | |
QBEWRQHVWMGSDD
|
7.0 | IC50 | 3 | — | |
QBGWTIGNWJPBDT
|
7.0 | IC50 | 3 | — | |
QBQRMCAZZBIYEL
|
7.0 | IC50 | 3 | — | |
QBUBVSIDQUINRB
|
7.0 | IC50 | 3 | — | |
QDMPTXGINYJNAN
|
7.0 | IC50 | 3 | — | |
QDSFQQGJJWMPBG
|
7.0 | IC50 | 3 | — | |
QGQSFDGKZWNNPG
|
7.0 | IC50 | 2 | — | |
QHPHQQAAAGTPSO
|
7.0 | IC50 | 3 | — | |
QJPBWDTZYARJRG
|
7.0 | IC50 | 2 | — | |
QNURCIHOTNZHID
|
7.0 | IC50 | 3 | — | |
QOBXXWBQZMXLLJ
|
7.0 | IC50 | 3 | — | |
QUKZLAGNAUMHTC
|
7.0 | IC50 | 3 | — | |
QWHVHAJJGFXJQO
|
7.0 | IC50 | 3 | — | |
QYULKCUUHHJJIU
|
7.0 | IC50 | 3 | — | |
QZGRYLFULFHDSH
|
7.0 | IC50 | 3 | — | |
RDOWVGMCRRFHTA
|
7.0 | IC50 | 2 | — | |
RLFHUVUKZFFZBK
|
7.0 | IC50 | 3 | — | |
RLJAGPBWFJHYAW
|
7.0 | IC50 | 3 | — | |
RMTHOSWPRSOFNF
|
7.0 | IC50 | 3 | — | |
RPTRIRFDPKDZCT
|
7.0 | IC50 | 3 | — | |
RQQVGERZDQNWTK
|
7.0 | IC50 | 2 | — | |
RRBNREHEKNKYJD
|
7.0 | IC50 | 2 | — | |
RSPAFCYZCBCSLK
|
7.0 | IC50 | 3 | — | |
RYEFRTKTDGXOLK
|
7.0 | IC50 | 3 | — | |
RZOXRAQOJQKDEH
|
7.0 | IC50 | 3 | — | |
RZQUJJFZDJNOMH
|
7.0 | IC50 | 3 | — | |
SATXBUGSMHGDCG
|
7.0 | IC50 | 2 | — | |
SBIZGGYJXGYHQC
|
7.0 | IC50 | 2 | — | |
SDVPFBNIPJXMAA
|
7.0 | IC50 | 3 | — | |
SJSLVLWUSQSVDO
|
7.0 | IC50 | 2 | — | |
SKLPIVFTLJZCBW
|
7.0 | IC50 | 2 | — | |
SLQAEOCZMOGNPB
|
7.0 | IC50 | 2 | — | |
SNWKZGWMPRZQQN
|
7.0 | IC50 | 3 | — | |
SQSZOQJFYXAWHR
|
7.0 | IC50 | 3 | — | |
SSTMRAVQPNLFAK
|
7.0 | IC50 | 3 | — | |
SUFPCLCMLRGXFH
|
7.0 | IC50 | 3 | — | |
SUNCVSGYFLTRPO
|
7.0 | IC50 | 3 | — | |
SVQYLXMEIGEJFO
|
7.0 | IC50 | 3 | — | |
SVSOFLSVCDVJQQ
|
7.0 | IC50 | 3 | — | |
SWBMRWPZBXKGLL
|
7.0 | IC50 | 3 | — | |
TUFZSBCXUZRADO
|
7.0 | IC50 | 2 | — |