Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KHINBPDUCGVKPG
|
7.0 | IC50 | 3 | — | |
KIKQCMFHJBBLPO
|
7.0 | IC50 | 2 | — | |
KMLOSXVUWJQNDP
|
7.0 | IC50 | 3 | — | |
KSCJDMZOEHAJSS
|
7.0 | IC50 | 2 | — | |
KSXPMSDQFDBYSH
|
7.0 | IC50 | 3 | — | |
KYRHLFLRSKNTMY
|
7.0 | IC50 | 3 | — | |
KYZMDLZMTIIYOU
|
7.0 | IC50 | 3 | — | |
LHUMLHFISNDFEG
|
7.0 | IC50 | 3 | — | |
LKLZCWIIVIPJTM
|
7.0 | IC50 | 3 | — | |
LNLAVZYUZRIWTM
|
7.0 | IC50 | 3 | — | |
LNRDHEBUMQFPKX
|
7.0 | IC50 | 2 | — | |
LPTUNCPXCKVCNQ
|
7.0 | IC50 | 2 | — | |
LPZUVSPPQUFWSE
|
7.0 | IC50 | 3 | — | |
LSPSSKVZRRFTTL
|
7.0 | IC50 | 2 | — | |
LSWGKRCLMQERHK
|
7.0 | IC50 | 3 | — | |
LTRMTOJBCQKBEH
|
7.0 | IC50 | 3 | — | |
LUCILDQKERZJEB
|
7.0 | IC50 | 3 | — | |
LYUZANVMMLWOOG
|
7.0 | IC50 | 3 | — | |
LZJGSIHOIRPDBW
|
7.0 | IC50 | 3 | — | |
LZNUJWUOFQBZEX
|
7.0 | IC50 | 2 | — | |
MGBWTZFJARAUGC
|
7.0 | IC50 | 3 | — | |
MGEROXNTVPRSKZ
|
7.0 | IC50 | 3 | — | |
MICBUWWORPLJCV
|
7.0 | IC50 | 3 | — | |
MIUDBUOGVNTIMI
|
7.0 | IC50 | 3 | — | |
MLKBCXWIKNAMOJ
|
7.0 | IC50 | 3 | — | |
MQSAEDIRZPBUJM
|
7.0 | IC50 | 3 | — | |
MREUVPMNGLXQLH
|
7.0 | IC50 | 3 | — | |
MSGCTRGQGAXORW
|
7.0 | IC50 | 3 | — | |
MWGVFCZWZWMNFV
|
7.0 | IC50 | 3 | — | |
MXMUBEMTNXLXIU
|
7.0 | IC50 | 3 | — | |
MZSYPKUZWGIZDW
|
7.0 | IC50 | 3 | — | |
NCWAELYKFLAQHW
|
7.0 | IC50 | 2 | — | |
NEEWJLXKBCBIGB
|
7.0 | IC50 | 3 | — | |
NFFHPPZZFWJGSH
|
7.0 | IC50 | 3 | — | |
NFKWWGSDAMVUAT
|
7.0 | IC50 | 3 | — | |
NHQHROKXXUCMLE
|
7.0 | IC50 | 3 | — | |
NIGMHJHMCSAYFE
|
7.0 | IC50 | 3 | — | |
NLTFQLISTSUENC
|
7.0 | IC50 | 3 | — | |
NYJCLYDJCHIMFW
|
7.0 | IC50 | 3 | — | |
OETMLVRYFJWGAX
|
7.0 | IC50 | 3 | — | |
OFJLEAIINHDRSW
|
7.0 | IC50 | 3 | — | |
OKFXEFRSSDSOQW
|
7.0 | IC50 | 3 | — | |
OOKUDGPQVOVZTN
|
7.0 | IC50 | 3 | — | |
OOLPARUANSTKCI
|
7.0 | IC50 | 3 | — | |
OTUJLGHUPZWNTF
|
7.0 | IC50 | 3 | — | |
OVPGPUIOPKYMQR
|
7.0 | IC50 | 2 | — | |
OYRAZNGOSIVXEX
|
7.0 | IC50 | 3 | — | |
OZPLGIFSKDBUEU
|
7.0 | IC50 | 3 | — | |
PECBVAQTPPRVRB
|
7.0 | IC50 | 3 | — | |
PGSMJKGDWYOKBQ
|
7.0 | IC50 | 3 | — |