Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DAAMUEUKNPYRPI
|
7.0 | IC50 | 3 | — | |
DELPLUDVOWJATI
|
7.0 | IC50 | 3 | — | |
DGMRHQKRWURCMX
|
7.0 | IC50 | 3 | — | |
DGRKTLAGZQDZKT
|
7.0 | IC50 | 3 | — | |
DIHHXPKERFBTAH
|
7.0 | IC50 | 3 | — | |
DOKMDLZQSRWMHM
|
7.0 | IC50 | 3 | — | |
DSCTUDBLSXZIJA
|
7.0 | IC50 | 3 | — | |
DWHYLPGLRMHNLA
|
7.0 | IC50 | 3 | — | |
DYZKDBCXQPHYOW
|
7.0 | IC50 | 3 | — | |
FCDUJXCEQMONRT
|
7.0 | IC50 | 3 | — | |
FCQKKNPJIZSOFM
|
7.0 | IC50 | 3 | — | |
FEMNETXMVKEMJZ
|
7.0 | IC50 | 2 | — | |
FEOPAGLTWFBXPN
|
7.0 | IC50 | 2 | — | |
FGTLXOSYVWGYEE
|
7.0 | IC50 | 2 | — | |
FMYGFJXXTNSQML
|
7.0 | IC50 | 3 | — | |
FMYGFJXXTNSQML
|
7.0 | IC50 | 3 | — | |
FOUBATKNDZVYKQ
|
7.0 | IC50 | 3 | — | |
FQALIHGLVDVIMA
|
7.0 | IC50 | 3 | — | |
FSMPTVIKNHGGJO
|
7.0 | IC50 | 3 | — | |
FSTPKVAGHDPQOZ
|
7.0 | IC50 | 3 | — | |
FXXYSJGZNUHXTP
|
7.0 | IC50 | 3 | — | |
FYRDJBHIWMIOQS
|
7.0 | IC50 | 3 | — | |
FZTYPXUSWRKGQD
|
7.0 | IC50 | 3 | — | |
GHQLSQHPXBFWCR
|
7.0 | IC50 | 3 | — | |
GICYOAGGKVTALK
|
7.0 | IC50 | 3 | — | |
GKKZRQXWOXFPPU
|
7.0 | IC50 | 2 | — | |
GOVSUZAVRQJORD
|
7.0 | IC50 | 3 | — | |
GTQJVOUAINIUPY
|
7.0 | IC50 | 2 | — | |
GUOCEPTXKXOBGI
|
7.0 | IC50 | 3 | — | |
GYYFJDQIMURKAF
|
7.0 | IC50 | 3 | — | |
HCNFOYIEZHCOME
|
7.0 | IC50 | 3 | — | |
HFAUCQJESVUACL
|
7.0 | IC50 | 3 | — | |
HLRYJUPVRHUTFL
|
7.0 | IC50 | 3 | — | |
HTDHJSKYCQHNPJ
|
7.0 | IC50 | 3 | — | |
HVOHDOQIFVGTOE
|
7.0 | IC50 | 2 | — | |
HXKZMHDDBKSOTA
|
7.0 | IC50 | 3 | — | |
IAXMOSJINXJMPE
|
7.0 | IC50 | 3 | — | |
IDBPBYMGBNZBKM
|
7.0 | IC50 | 3 | — | |
IEXXFYGUTSBWAA
|
7.0 | IC50 | 3 | — | |
IIILCAYWUVJASR
|
7.0 | IC50 | 3 | — | |
ILHBWUSIWJTAFW
|
7.0 | IC50 | 3 | — | |
IMRPCULDPOGBFT
|
7.0 | IC50 | 3 | — | |
INNUGJACJWCMHU
|
7.0 | IC50 | 3 | — | |
IVWCPGWFHKHDGS
|
7.0 | IC50 | 3 | — | |
IXBGWFGVYLAJRO
|
7.0 | IC50 | 3 | — | |
JBZXPIPNDSVIOW
|
7.0 | IC50 | 3 | — | |
JLMDPBMMFGTSPS
|
7.0 | IC50 | 3 | — | |
JMTDZCXJUVRYOX
|
7.0 | IC50 | 3 | — | |
JSEPPFHHSFLYAV
|
7.0 | IC50 | 2 | — | |
KFJSDJBSMAFDTM
|
7.0 | IC50 | 3 | — |