Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
COLQRVWEVUYXEE
|
7.0 | IC50 | 2 | — | |
MKXRYOOPYMOGHI
|
7.0 | IC50 | 2 | — | |
RWOFWISHLYBHDE
|
7.0 | IC50 | 2 | — | |
YCXZBULDUGDETC
|
7.0 | IC50 | 2 | — | |
YXLDQBFWFZDCOF
|
7.0 | IC50 | 3 | — | |
BOTRGRDIRVJRGQ
|
7.0 | IC50 | 2 | — | |
KXMZDGSRSGHMMK
|
7.0 | IC50 | 14 | — | |
YCGFHHACUCVQPI
|
7.0 | IC50 | 2 | — | |
BNEVROJYJXVARX
|
7.0 | IC50 | 2 | — | |
GAZFCMBOTHVCNP
|
7.0 | IC50 | 2 | — | |
SNSHWVBULOTYEY
|
7.0 | IC50 | 3 | — | |
UDHIJSWGTJKLCI
|
7.0 | IC50 | 2 | — | |
WZIASJJBXMZPDE
|
7.0 | IC50 | 2 | — | |
YCGFHHACUCVQPI
|
7.0 | IC50 | 2 | — | |
FVPWCMRDQTVHGA
|
7.0 | IC50 | 2 | — | |
KFASJVNZRIDONN
|
7.0 | IC50 | 2 | — | |
JIUGKBKCSODYEF
|
7.0 | IC50 | 2 | — | |
NXSJMRCTGYTSTK
|
7.0 | Kd | 200 | — | |
OSVUGUHRKMMBSE
|
7.0 | Kd | 170 | — | |
WFHGEWDDDBUGKR
|
7.0 | IC50 | 2 | — | |
AAAVFZXQZLILOV
|
7.0 | IC50 | 2 | — | |
AETSJLUJNHRHTF
|
7.0 | IC50 | 3 | — | |
AEZKBVGBJHBFSN
|
7.0 | IC50 | 3 | — | |
AFPSKIHTKZXBFT
|
7.0 | IC50 | 3 | — | |
APBVBNCCTNJHNI
|
7.0 | IC50 | 3 | — | |
ASMRZAURCVEUDT
|
7.0 | IC50 | 3 | — | |
AYGHFYGVUSZIQX
|
7.0 | IC50 | 3 | — | |
BAPMAEPDSGOVLW
|
7.0 | IC50 | 3 | — | |
BCXFNEUUCDUFKI
|
7.0 | IC50 | 3 | — | |
BFNFLZYHFBADOM
|
7.0 | IC50 | 3 | — | |
BHKWLDYFVDSONJ
|
7.0 | IC50 | 3 | — | |
BIJDJWLTYUZFKL
|
7.0 | IC50 | 3 | — | |
BNPDEZXLADUGPG
|
7.0 | IC50 | 3 | — | |
BODQMNJDMPCWJG
|
7.0 | IC50 | 3 | — | |
BPJMLEPJLRDHSW
|
7.0 | IC50 | 2 | — | |
BPWQOFIOJRRAHB
|
7.0 | IC50 | 3 | — | |
BRRFZOMLPLZBEN
|
7.0 | IC50 | 3 | — | |
BTXCTSVHJPQIOO
|
7.0 | IC50 | 3 | — | |
CAHKFKZSJNQNFZ
|
7.0 | IC50 | 3 | — | |
CAWNAGGQKYMUOR
|
7.0 | IC50 | 3 | — | |
CCHKPKLVTJIEKB
|
7.0 | IC50 | 3 | — | |
CDPWYOOXYRMDFM
|
7.0 | IC50 | 2 | — | |
CEABUWJXZBOYLD
|
7.0 | IC50 | 3 | — | |
CEGMNUFOCROAKS
|
7.0 | IC50 | 3 | — | |
CFZJCRMOAAJBIX
|
7.0 | IC50 | 3 | — | |
CIQGHNQVQGZPKP
|
7.0 | IC50 | 3 | — | |
CKIJILKJTWPRNY
|
7.0 | IC50 | 3 | — | |
CPIJQYGEORDTME
|
7.0 | IC50 | 3 | — | |
CPKPERZPHDRHKD
|
7.0 | IC50 | 3 | — | |
CRCJXGPYZWLPSL
|
7.0 | IC50 | 3 | — |