Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KYCKKSZMVINEPM
|
9.0 | IC50 | 4 | — | |
LOLPPWBBNUVNQZ
|
9.0 | IC50 | 97 | Yes | |
OUJHQVBNJZKTSS
|
9.0 | IC50 | 2 | — | |
UOIRCOJSMABXQO
|
9.0 | IC50 | 2 | — | |
VNPYBQLMWOYRMR
|
9.0 | IC50 | 4 | — | |
YOXIVEDZDMDJSA
|
9.0 | IC50 | 3 | — | |
YSCRAUWGPPUZRI
|
9.0 | IC50 | 4 | — | |
DNXCFFPPWFGXKA
|
9.0 | IC50 | 3 | — | |
AAUNIEBMIUGNTA
|
9.0 | IC50 | 4 | — | |
AGIHELYBRFIVHZ
|
9.0 | IC50 | 4 | — | |
CWFMWJSSAAOUBO
|
9.0 | IC50 | 4 | — | |
KAAPXWSYROPAEL
|
9.0 | IC50 | 4 | — | |
MJSHVHLADKXCML
|
9.0 | IC50 | 4 | — | |
NEZRLVDPFUFEKB
|
9.0 | IC50 | 3 | — | |
NEZRLVDPFUFEKB
|
9.0 | IC50 | 4 | — | |
UEMPFKOYBHCUIG
|
9.0 | IC50 | 4 | — | |
VEFDEIILCRXHNC
|
9.0 | IC50 | 4 | — | |
BBJHTTNJKZUZCD
|
8.9 | IC50 | 4 | — | |
BTHRAPVJUCSEGQ
|
8.9 | IC50 | 4 | — | |
BVIDZAGIDOQWSF
|
8.9 | IC50 | 4 | — | |
CDPXZDPKRHLKCH
|
8.9 | IC50 | 4 | — | |
FXPKSABYJKCHOV
|
8.9 | IC50 | 4 | — | |
NBIOGGWEVWYBFI
|
8.9 | IC50 | 4 | — | |
YAUQWMBRTAHSFI
|
8.9 | IC50 | 4 | — | |
AVQBNZOTTBHSCI
|
8.9 | IC50 | 4 | — | |
CKRMOFCKEANQCR
|
8.9 | IC50 | 4 | — | |
DWFDADABQIDXBP
|
8.9 | IC50 | 4 | — | |
HTMNAROLUQALML
|
8.9 | IC50 | 4 | — | |
LBEJYFVJIPQSNX
|
8.9 | IC50 | 4 | — | |
PRABTKJJUJZVNX
|
8.9 | IC50 | 4 | — | |
PWOIRDUWFWWFMT
|
8.9 | IC50 | 4 | — | |
PWOIRDUWFWWFMT
|
8.9 | IC50 | 3 | — | |
QXQKUTDAZQEITC
|
8.9 | IC50 | 4 | — | |
RGJASBGADDXMBE
|
8.9 | IC50 | 4 | — | |
YLAIGAIPEXSTTK
|
8.9 | IC50 | 3 | — | |
DCSJNPUSJYLHBA
|
8.8 | IC50 | 3 | — | |
IKENQUDOTQBCJH
|
8.8 | Kd | 18 | — | |
NDWOEUVAOGUXGP
|
8.8 | IC50 | 4 | — | |
VUZLNWIIHACTEC
|
8.8 | IC50 | 4 | — | |
VXVHXDKIVTYZHG
|
8.8 | IC50 | 2 | — | |
VZHCQBXYACZHPJ
|
8.8 | IC50 | 3 | — | |
ZSQUNKBTVLUHTH
|
8.8 | IC50 | 2 | — | |
AIIRAHKUAWNOHT
|
8.8 | IC50 | 2 | — | |
CRJMKZAXSRYICG
|
8.8 | IC50 | 2 | — | |
DHCWIUCAJNMGDF
|
8.8 | IC50 | 4 | — | |
QQTWEWAFAIDGJB
|
8.8 | IC50 | 4 | — | |
RCQLJPMEVONOSW
|
8.8 | IC50 | 4 | — | |
UMJNEGIWFHRTLO
|
8.8 | IC50 | 4 | — | |
BPKUEQDPPXTOSG
|
8.8 | IC50 | 4 | — | |
BSDOEKCQNXKTDO
|
8.8 | IC50 | 2 | — |