Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IPHZKBACASVMHL
|
7.2 | IC50 | 2 | — | |
ONOSFELSQUOGIC
|
7.2 | IC50 | 3 | — | |
QQGGOMPVIRZWRW
|
7.2 | IC50 | 2 | — | |
RBGWDTGTACCPGE
|
7.2 | IC50 | 2 | — | |
WAHPBOBQSDMVRH
|
7.2 | IC50 | 2 | — | |
WHCPVMMPHZOQIK
|
7.2 | IC50 | 3 | — | |
YHEINTAUSLSCDI
|
7.2 | IC50 | 3 | — | |
YQBNFYFUPHSRMR
|
7.2 | IC50 | 3 | — | |
CTNPALGJUAXMMC
|
7.2 | Kd | 151 | — | |
ISPBCAXOSOLFME
|
7.2 | IC50 | 11 | — | |
RQAATFYANFZYNJ
|
7.2 | IC50 | 2 | — | |
SPERNPFVNHOOND
|
7.2 | IC50 | 2 | — | |
AZIQVRPNDXMEOX
|
7.2 | IC50 | 2 | — | |
BPDHUCWPIWLNQJ
|
7.2 | IC50 | 2 | — | |
KHCNBZBQEJGAOZ
|
7.2 | IC50 | 2 | — | |
PQSZJQKHNTZKEY
|
7.2 | IC50 | 2 | — | |
ZRODNORXCGXTQW
|
7.2 | IC50 | 2 | — | |
CNDSIFCMFBHBNW
|
7.1 | IC50 | 2 | — | |
FAILDDCVKDFVJQ
|
7.1 | IC50 | 2 | — | |
GZYCQQBRSRIFII
|
7.1 | Kd | 7 | — | |
HVIDXJFXDHKCMO
|
7.1 | IC50 | 4 | — | |
MMOZHTDOCYODPM
|
7.1 | IC50 | 4 | — | |
MXNSTJDJNSFMJJ
|
7.1 | IC50 | 3 | — | |
WZXCBFSKSWUTOQ
|
7.1 | IC50 | 2 | — | |
XVJQKOIBNAWHNV
|
7.1 | IC50 | 2 | — | |
AYJMUFFYIOWRRM
|
7.1 | IC50 | 2 | — | |
BSMUSWHXZAXDID
|
7.1 | IC50 | 3 | — | |
CMWRPDHVGMHLSZ
|
7.1 | IC50 | 22 | — | |
ATNVOCQRWNYCHO
|
7.1 | IC50 | 2 | — | |
GFZCTGHGFMTANV
|
7.1 | IC50 | 2 | — | |
MXNSTJDJNSFMJJ
|
7.1 | IC50 | 2 | — | |
WYWDFLXMMGKGOW
|
7.1 | IC50 | 4 | — | |
ASMYWCGHYWQPGO
|
7.1 | IC50 | 4 | — | |
JHFPXAGOMRSTRG
|
7.1 | IC50 | 2 | — | |
QZIANMAYEYYSQX
|
7.1 | IC50 | 2 | — | |
ADLLAPNUCPCMFE
|
7.1 | IC50 | 2 | — | |
PUZKUEMWVFYLJR
|
7.1 | IC50 | 3 | — | |
CDNSOMCMTZMHON
|
7.1 | IC50 | 3 | — | |
FPQXIYKYKQSXAR
|
7.1 | IC50 | 2 | — | |
GUBJNPWVIUFSTR
|
7.1 | Kd | 103 | — | |
NUBZRIXZYLGEIM
|
7.1 | IC50 | 2 | — | |
UKYJKXMPIDEQFF
|
7.1 | IC50 | 16 | — | |
XXEJLOWSXIMQHG
|
7.1 | IC50 | 4 | — | |
WPBQHEXHVOGJHS
|
7.1 | IC50 | 2 | — | |
YLHVXJHQPQYBSW
|
7.1 | IC50 | 2 | — | |
ZNORSSZINYHFFL
|
7.1 | IC50 | 2 | — | |
HJFLVMBTWIJCNF
|
7.0 | IC50 | 3 | — | |
LBFYYFRPBFRKSE
|
7.0 | IC50 | 2 | — | |
XCXMZUYZFOFSTB
|
7.0 | IC50 | 2 | — | |
AKWLDQDWZNJYKL
|
7.0 | IC50 | 14 | — |